Berek Novak's Gyn 2019. Chapter 7. Reproductive Physiology

 Reproductive Physiology

BS. Nguyễn Hồng Anh

KEY POINTS

1 The female reproductive process involves the central nervous system (primarily

hypothalamus), the pituitary gland, the ovary, and the uterus (endometrium). All

must function appropriately for normal reproduction to occur.

2 Hypothalamic gonadotropin-releasing hormone (GnRH) simultaneously regulates the

luteinizing hormone (LH) and follicle-stimulating hormone (FSH) in the pituitary

through pulsatile secretions. The pulse frequency determines the relative amounts of

LH and FSH secretion.

3 The ovary responds to FSH and LH in a defined, sequential manner to produce

follicular growth, ovulation, and corpus luteum formation. The cycle is designed to

produce an optimal environment for pregnancy; if pregnancy does not occur, the

cycle begins again.

4 In the early menstrual cycle the ovary produces estrogen, which is responsible for

endometrial growth. After ovulation, progesterone is produced in significant

quantities, which transforms the endometrium into a form ideal for implantation of

the embryo. If no pregnancy occurs, the ovary ceases to produce estrogen and

progesterone, the endometrium is sloughed, and the cycle repeats.

[1] The reproductive process in women is a complex and highly evolved

interaction of many components. The carefully orchestrated series of events that

contributes to a normal ovulatory menstrual cycle requires precise timing and

regulation of hormonal input from the central nervous system (CNS), pituitary

gland, and ovary. This delicately balanced process can be disrupted easily and

result in reproductive failure, which is a major clinical issue confronting

gynecologists. To manage such conditions effectively, it is critical that

gynecologists understand the normal physiology of the menstrual cycle. The

anatomic structures, hormonal components, and their interactions, play a vital role

in the function of the reproductive system. Fitting together the various pieces of

this intricate puzzle creates “the big picture”: an overview of how the

reproductive system of women is designed to function.

NEUROENDOCRINOLOGY

Neuroendocrinology represents facets of two traditional fields of medicine:

endocrinology, which is the study of hormones (i.e., substances secreted into the

bloodstream that have diverse actions at sites remote from the point of secretion);

and neuroscience, which is the study of the action of neurons. The discovery of

neurons that transmit impulses and secrete their products into the vascular system

283to function as hormones, a process known as neurosecretion, demonstrates that

the two systems are intimately linked. For instance, the menstrual cycle is

regulated through the feedback of hormones on the neural tissue of the CNS.

ANATOMY

Hypothalamus

The hypothalamus is a small neural structure situated at the base of the

brain above the optic chiasm and below the third ventricle (Fig. 7-1). It is

connected directly to the pituitary gland and is the part of the brain that is

the source of many pituitary secretions. Anatomically, the hypothalamus is

divided into three zones: periventricular (adjacent to the third ventricle); medial

(primarily cell bodies); and lateral (primarily axonal). Each zone is further

subdivided into structures known as nuclei, which represent locations of

concentrations of similar types of neuronal cell bodies (Fig. 7-2).

284FIGURE 7-1 The hypothalamus and its neurologic connections to the pituitary.

285FIGURE 7-2 The neuronal cell bodies of the hypothalamus.

The hypothalamus is not an isolated structure within the CNS; instead, it

has multiple interconnections with other regions in the brain. In addition to

the well-known pathways of hypothalamic output to the pituitary, there are

numerous less well-characterized pathways of output to diverse regions of the

brain, including the limbic system (amygdala and hippocampus), the thalamus,

and the pons (1). Many of these pathways form feedback loops to areas supplying

neural input to the hypothalamus.

286287FIGURE 7-3 The hypothalamic secretory products function as pituitary-releasing factors

that control the endocrine function of the ovaries, the thyroid, and the adrenal glands.

CRH, corticotropin releasing hormone; TRH, thyrotropin releasing hormone; GnRH,

gonadotropin releasing hormone; FSH, follicle stimulating hormone; LH, leutinizing

hormone; T4, thyroxine; ACTH, adrenocorticotropic hormone; TSH, thyroid stimulating

hormone; and E2, estradiol.

Several levels of feedback to the hypothalamus exist and are known as the

long, short, and ultrashort feedback loops. The long feedback loop is

composed of endocrine input from circulating hormones, just as is the feedback of

androgens and estrogens onto steroid receptors in the hypothalamus (2,3).

Similarly, pituitary hormones may feed back to the hypothalamus and serve

important regulatory functions in short-loop feedback. Finally, hypothalamic

secretions may directly feed back to the hypothalamus itself in an ultrashort

feedback loop.

The major secretory products of the hypothalamus are the pituitaryreleasing factors (Fig. 7-3):

1. Gonadotropin-releasing hormone (GnRH), which controls the secretion of

luteinizing hormone (LH) and follicle-stimulating hormone (FSH)

2. Corticotropin-releasing hormone (CRH), which controls the release of

adrenocorticotrophic hormone (ACTH)

3. Growth hormone–releasing hormone (GHRH), which regulates the release

of growth hormone (GH)

4. Thyrotropin-releasing hormone (TRH), which regulates the secretion of

thyroid-stimulating hormone (TSH)

The hypothalamus is the source of all neurohypophyseal hormone

production. The neural posterior pituitary can be viewed as a direct extension of

the hypothalamus connected by the finger-like infundibular stalk. The capillaries

in the median eminence differ from those in other regions of the brain. Unlike the

usual tight junctions that exist between adjacent capillary endothelial lining cells,

the capillaries in this region are fenestrated in the same manner as capillaries

outside the CNS. As a result, there is no blood–brain barrier in the median

eminence.

Pituitary

The pituitary is divided into three regions or lobes: anterior, intermediate, and

posterior. The anterior pituitary (adenohypophysis) is quite different structurally

from the posterior neural pituitary (neurohypophysis), which is a direct physical

288extension of the hypothalamus. The adenohypophysis is derived embryologically

from epidermal ectoderm from an infolding of Rathke pouch. Therefore, it is not

composed of neural tissue, as is the posterior pituitary, and does not have direct

neural connections to the hypothalamus. Instead, a unique anatomic relationship

exists that combines elements of neural production and endocrine secretion.

The adenohypophysis itself has no direct arterial blood supply. Its major source

of blood flow is also its source of hypothalamic input—the portal vessels. Blood

flow in these portal vessels is primarily from the hypothalamus to the pituitary.

Blood is supplied to the posterior pituitary via the superior, middle, and inferior

hypophyseal arteries. In contrast, the anterior pituitary has no direct arterial blood

supply. Instead, it receives blood via a rich capillary plexus of the portal vessels

that originates in the median eminence of the hypothalamus and descends along

the pituitary stalk. This pattern is not absolute, however, and retrograde blood

flow has occurred (4). This blood flow, combined with the location of the median

eminence outside the blood–brain barrier, permits bidirectional feedback control

between the two structures.

The specific secretory cells of the anterior pituitary are classified based on

their hematoxylin- and eosin-staining patterns. Acidophilic-staining cells

primarily secrete GH and prolactin and, to a variable degree, ACTH (5). The

gonadotropins are secreted by basophilic cells, and TSH is secreted by the

neutral-staining chromophobes.

REPRODUCTIVE HORMONES

Hypothalamus

Gonadotropin-Releasing Hormone

GnRH (also called luteinizing hormone–releasing hormone, or LHRH) is the

controlling factor for gonadotropin secretion (6). It is a decapeptide produced

by neurons with cell bodies primarily in the arcuate nucleus of the hypothalamus

(7–9) (Fig. 7-4). Embryologically, these neurons originate in the olfactory pit and

migrate to their adult locations (10). These GnRH-secreting neurons project axons

that terminate on the portal vessels at the median eminence where GnRH is

secreted for delivery to the anterior pituitary. Less clear in function are multiple

other secondary projections of GnRH neurons to locations within the CNS.

The gene that encodes GnRH produces a 92-amino-acid precursor protein,

which contains the GnRH decapeptide and a 56 amino acid peptide known as

GnRH-associated peptide (GAP). The GAP is a potent inhibitor of prolactin

secretion and a stimulator of gonadotropin release.

Pulsatile Secretion

289[2] GnRH is unique among releasing hormones in that it simultaneously

regulates the secretion of two hormones—FSH and LH. It is unique among

the body’s hormones because it must be secreted in a pulsatile fashion to be

effective, and the pulsatile release of GnRH influences the release of the two

gonadotropins (11–13). Using animals that had undergone electrical

destruction of the arcuate nucleus and had no detectable levels of

gonadotropins, a series of experiments were performed with varying dosages

and intervals of GnRH infusion (13,14). Continual infusions did not result in

gonadotropin secretion, whereas a pulsatile pattern led to physiologic

secretion patterns and follicular growth. Continual exposure of the pituitary

gonadotroph to GnRH results in a phenomenon calleddownregulation,

through which the number of gonadotroph cell surface GnRH receptors is

decreased (15). Similarly, intermittent exposure to GnRH will “upregulate”

or “autoprime” the gonadotroph to increase its number of GnRH receptors

(16). This allows the cell to have a greater response to subsequent GnRH

exposure. Similar to the intrinsic electrical pacemaker cells of the heart, this

action most likely represents an intrinsic property of the GnRH-secreting neuron,

although it is subject to modulation by various neuronal and hormonal inputs to

the hypothalamus.

The continual pulsatile secretion of GnRH is necessary because GnRH has

an extremely short half-life (only 2 to 4 minutes) as a result of rapid

proteolytic cleavage. The pulsatile secretion of GnRH varies in frequency and

amplitude throughout the menstrual cycle and is tightly regulated (Fig. 7-5)

(17,18).

The follicular phase is characterized by frequent, small-amplitude pulses of

GnRH secretion. In the late follicular phase, there is an increase in frequency and

amplitude of pulses. During the luteal phase, however, there is a progressive

lengthening of the interval between pulses. The amplitude in the luteal phase is

higher than that in the follicular phase, but it declines progressively over the 2

weeks. This variation in pulse frequency allows for variation in LH and FSH

throughout the menstrual cycle. For example, decreasing the pulse frequency of

GnRH decreases LH secretion but increases FSH, an important aspect of

enhancing FSH availability in the late luteal phase. The pulse frequency is not the

sole determinant of pituitary response; additional hormonal influences, such as

those exerted by ovarian peptides and sex steroids, can modulate the GnRH

effect.

290FIGURE 7-4 Gonadotropin-releasing hormone is a decapeptide.

FIGURE 7-5 The pulsatile secretion of gonadotropin-releasing hormone in the follicular

and luteal phases of the cycle.

Although GnRH is primarily involved in endocrine regulation of

gonadotropin secretion from the pituitary, it is apparent that this molecule

has autocrine and paracrine functions throughout the body. The decapeptide

is found in neural and nonneural tissues; receptors are present in many

extrapituitary structures, including the ovary and placenta. Data suggest that

291GnRH may be involved in regulating human chorionic gonadotropin (hCG)

secretion and implantation, and in decreasing cell proliferation and mediating

apoptosis in tumor cells (19). The role of GnRH in the extrapituitary sites remains

to be fully elucidated.

Gonadotropin-Releasing Hormone Agonists

Mechanism of Action

Used clinically, GnRH agonists are modifications of the native molecule to either

increase receptor affinity or decrease degradation (20). Their use leads to a

persistent activation of GnRH receptors, as if continuous GnRH exposure existed.

As would be predicted by the constant GnRH infusion experiments, this leads to

suppression of gonadotropin secretion. An initial release of gonadotropins is

followed by a profound suppression of secretion. The initial release of

gonadotropins represents the secretion of pituitary stores in response to receptor

binding and activation. With continued activation of the gonadotroph GnRH

receptor, however, there is a downregulation effect and a decrease in the

concentration of GnRH receptors. As a result, gonadotropin secretion decreases

and sex steroid production falls to castrate levels (21).

Additional modification of the GnRH molecule results in an analogue that

has no intrinsic activity but competes with GnRH for the same receptor site

(22). These GnRH antagonists produce a competitive blockade of GnRH

receptors, preventing stimulation by endogenous GnRH and causing an

immediate fall in gonadotropin and sex steroid secretion (23). The clinical

effect is observed within 24 to 72 hours. Moreover, antagonists may not function

solely as competitive inhibitors; evidence suggests they may also produce

downregulation of GnRH receptors, further contributing to the loss of

gonadotropin activity (24).

Structure—Agonists and Antagonists

As a peptide hormone, GnRH is degraded by enzymatic cleavage of bonds

between its amino acids. Pharmacologic alterations of the structure of GnRH led

to the creation of agonists and antagonists (Fig. 7-4). The primary sites of

enzymatic cleavage are between amino acids 5 and 6, 6 and 7, and 9 and 10.

Substitution of the position-6 amino acid glycine with large bulky amino acid

analogues makes degradation more difficult and creates a form of GnRH with a

relatively long half-life. Substitution at the carboxyl terminus produces a form of

GnRH with increased receptor affinity. The resulting high affinity and slow

degradation produces a molecule that mimics continuous exposure to native

GnRH (20). Thus, as with constant GnRH exposure, downregulation occurs.

GnRH agonists are widely used to treat disorders that are dependent on ovarian

292hormones (21). They are used to control ovulation induction cycles and treat

precocious puberty, ovarian hyperandrogenism, leiomyomas, endometriosis, and

hormonally dependent cancers. The development of GnRH antagonists proved

more difficult because a molecule was needed that maintained the binding and

degradation resistance of agonists but failed to activate the receptor. Early

attempts involved modification of amino acids 1 and 2, as well as those

previously utilized for agonists. Commercial antagonists have structural

modifications at amino acids 1, 2, 3, 6, 8, and 10. The treatment spectrum is

expected to be similar to that of GnRH agonists, but with a more rapid onset of

action.

Nonpeptide, small molecule structures with high affinity for the GnRH receptor

were developed (25). These compounds demonstrated the ability to suppress the

reproductive axis in a dose-related manner via oral administration, unlike the

parenteral approach required with traditional peptide analogues (26). Investigation

may elucidate an expanded therapeutic role for these antagonists.

Endogenous Opioids and Effects on GnRH

The endogenous opioids are three related families of naturally occurring

substances produced in the CNS that represent the natural ligands for the opioid

receptors (27–29). There are three major classes of endogenous opioids, each

derived from precursor molecules:

1. Endorphins are named for their endogenous morphine-like activity. These

substances are produced in the hypothalamus from the precursor

proopiomelanocortin (POMC) and have diverse activities, including regulation

of temperature, appetite, mood, and behavior (30).

2. Enkephalins are the most widely distributed opioid peptides in the brain, and

they function primarily in regulation of the autonomic nervous system.

Proenkephalin A is the precursor for the two enkephalins of primary

importance: methionine–enkephalin and leucine–enkephalin.

3. Dynorphins are endogenous opioids produced from the precursor

proenkephalin B that serve a function similar to that of the endorphins,

producing behavioral effects and exhibiting a high analgesic potency.

The endogenous opioids play a significant role in the regulation of

hypothalamic–pituitary function. Endorphins appear to inhibit GnRH

release within the hypothalamus, resulting in inhibition of gonadotropin

secretion (31). Ovarian sex steroids can increase the secretion of central

endorphins, further depressing gonadotropin levels (32).

Endorphin levels vary significantly throughout the menstrual cycle, with

293peak levels in the luteal phase and a nadir during menses (33). This inherent

variability, although helping to regulate gonadotropin levels, may contribute to

cycle-specific symptoms experienced by ovulatory women. For example, the

dysphoria experienced by some women in the premenstrual phase of the cycle

may be related to a withdrawal of endogenous opiates (34). This theory is

bolstered by the finding that inhibition of opiate withdrawal by naltrexone

alleviates many premenstrual symptoms (35).

Pituitary Hormone Secretion

Anterior Pituitary

The anterior pituitary is responsible for the secretion of the major hormonereleasing factors—FSH, LH, TSH, and ACTH—and GH and prolactin. Each

hormone is released by a specific pituitary cell type.

Gonadotropins

The gonadotropins FSH and LH are produced by the anterior pituitary

gonadotroph cells and are responsible for ovarian follicular stimulation.

Structurally, there is great similarity between FSH and LH (Fig. 7-6). They

are glycoproteins that share identical α subunits and differ only in the structure of

their β subunits, which confer receptor specificity (36,37). The synthesis of the β

subunits is the rate-regulating step in gonadotropin biosynthesis (38). TSH and

placental hCG share identical α subunits with the gonadotropins. There are

several forms of each gonadotropin, which differ in carbohydrate content as a

result of posttranslation modification. The degree of modification varies with

steroid levels and is an important regulator of gonadotropin bioactivity.

Prolactin

Prolactin, a 198-amino-acid polypeptide secreted by the anterior pituitary

lactotroph, is the primary trophic factor responsible for the synthesis of milk

by the breast (39). Several forms of this hormone, which are named according to

their size and bioactivity, are normally secreted (40). Prolactin gene transcription

is principally stimulated by estrogen; other hormones promoting transcription are

TRH and a variety of growth factors.

294FIGURE 7-6 The structural similarity between follicle-stimulating hormone (FSH),

luteinizing hormone (LH), and thyroid-stimulating hormone (TSH). The α subunits are

identical, and the β subunits differ.

Prolactin secretion is under tonic inhibitory control by the hypothalamic

secretion of dopamine (41). Therefore, disease states characterized by decreased

dopamine secretion or any condition that interrupts transport of dopamine down

the infundibular stalk to the pituitary gland will result in increased synthesis of

prolactin. In this respect, prolactin is unique in comparison with all other pituitary

hormones: It is predominantly under tonic inhibition, and release of control

produces an increase in secretion. Clinically, increased prolactin levels are

associated with amenorrhea and galactorrhea, and hyperprolactinemia

should be suspected in any individual with symptoms of either of these

conditions.

Although prolactin appears to be primarily under inhibitory control,

many stimuli can elicit its release, including breast manipulation, drugs,

stress, exercise, and certain foods. Hormones that may stimulate prolactin

release include TRH, vasopressin, γ-aminobutyric acid (GABA), dopamine, β-

endorphin, vasoactive intestinal peptide (VIP), epidermal growth factor (EGF),

angiotensin II, estrogens, and possibly GnRH (42–46). The relative contributions

of these substances under normal conditions remain to be determined.

Thyroid-Stimulating Hormone, Adrenocorticotropic Hormone, and Growth Hormone

The other hormones produced by the anterior pituitary are TSH, ACTH,

and GH. TSH is secreted by the pituitary thyrotrophs in response to TRH.

As with GnRH, TRH is synthesized primarily in the arcuate nucleus of the

hypothalamus and is secreted into the portal circulation for transport to the

pituitary. In addition to stimulating TSH release, TRH is a major stimulus for the

295release of prolactin. TSH stimulates release of T3 and T4 from the thyroid gland,

which in turn has a negative feedback effect on pituitary TSH secretion.

Abnormalities of thyroid secretion (hyper- and hypothyroidism) are frequently

associated with ovulatory dysfunction as a result of diverse actions on the

hypothalamic–pituitary–ovarian axis (47).

Adrenocorticotrophic hormone is secreted by the anterior pituitary in

response to another hypothalamic-releasing factor, CRH, and stimulates the

release of adrenal glucocorticoids. Unlike the other anterior pituitary products,

ACTH secretion has a diurnal variation with an early morning peak and a late

evening nadir. As with the other pituitary hormones, ACTH secretion is

negatively regulated by feedback from its primary end product, which in this case

is cortisol.

The anterior pituitary hormone that is secreted in the greatest absolute

amount is GH. It is secreted in response to the hypothalamic-releasing factor,

GHRH, and by thyroid hormone and glucocorticoids. This hormone is secreted in

a pulsatile fashion but with peak release occurring during sleep. In addition to its

vital role in the stimulation of linear growth, GH plays a diverse role in

physiologic homeostasis. The hormone plays a role in bone mitogenesis, CNS

function (improved memory, cognition, and mood), body composition, breast

development, and cardiovascular function. It also affects insulin regulation and

acts anabolically. GH appears to have a role in the regulation of ovarian function,

although the degree to which it serves this role in normal physiology is unclear

(48).

Posterior Pituitary

Structure and Function

The posterior pituitary (neurohypophysis) is composed exclusively of neural

tissue and is a direct extension of the hypothalamus. It lies directly adjacent to

the adenohypophysis but is embryologically distinct, derived from an

invagination of neuroectodermal tissue in the third ventricle. Axons in the

posterior pituitary originate from neurons with cell bodies in two distinct regions

of the hypothalamus, the supraoptic and paraventricular nuclei, named for their

anatomic relationship to the optic chiasm and the third ventricle. Together these

two nuclei compose the hypothalamic magnocellular system. These neurons can

secrete their synthetic products directly from axonal boutons into the general

circulation to act as hormones. This is the mechanism of secretion of the

hormones of the posterior pituitary, oxytocin and arginine vasopressin (AVP).

Although this is the primary mode of release for these hormones, numerous other

secondary pathways were identified, including secretion into the portal

296circulation, intrahypothalamic secretion, and secretion into other regions of the

CNS (49).

In addition to the established functions of oxytocin and vasopressin, several

other diverse roles were suggested in animal models. These functions include

modulation of sexual activity and appetite, learning and memory consolidation,

temperature regulation, and regulation of maternal behaviors (50). In the human,

these neuropeptides were linked to social attachment (51–53). Receptor variants

for these two molecules were linked to the spectrum of autistic disorders,

suggesting that proper function of these two neuropeptides with their receptors is

required for positive group interactive behavior. This relationship is strengthened

by a strong association between altruistic behavior and the length of the AVP-1a

receptor promoter region (52,54). Complex human behaviors may be partially

governed by a relatively simple neuropeptide system. Continuing investigation

should help elucidate this physiology and potential therapeutic interventions.

Oxytocin

Oxytocin is a 9-amino-acid peptide primarily produced by the

paraventricular nucleus of the hypothalamus (Fig. 7-7). The primary function

of this hormone in humans is the stimulation of two specific types of muscular

contractions (Fig. 7-8). The first type, uterine muscular contraction, occurs during

parturition. The second type of muscular contraction regulated by oxytocin is

breast lactiferous duct myoepithelial contractions, which occur during the milk

letdown reflex. Oxytocin release may be stimulated by suckling, triggered by a

signal from nipple stimulation transmitted via thoracic nerves to the spinal cord

and then to the hypothalamus, where oxytocin is released in an episodic fashion

(48). Oxytocin release may be triggered by olfactory, auditory, and visual clues,

and may play a role in the conditioned reflex in nursing animals. Stimulation of

the cervix and vagina can cause significant release of oxytocin, which may trigger

reflex ovulation (the Ferguson reflex) in some species.

FIGURE 7-7 Oxytocin and arginine vasopressin (AVP) are 9-amino-acid peptides

produced by the hypothalamus. They differ in only two amino acids.

297FIGURE 7-8 Oxytocin stimulates muscular contractions of the uterus during parturition

and the breast lactiferous duct during the milk letdown reflex. Arginine vasopressin (AVP)

regulates circulating blood volume, pressure, and osmolality.

Arginine Vasopressin

Also known as antidiuretic hormone (ADH), AVP is the second major

secretory product of the posterior pituitary (Fig. 7-7). It is synthesized

primarily by neurons with cell bodies in the supraoptic nuclei (Fig. 7-8). Its major

298function is the regulation of circulating blood volume, pressure, and osmolality

(55). Specific receptors throughout the body can trigger the release of AVP.

Osmoreceptors located in the hypothalamus sense changes in blood osmolality

from a mean of 285 mOsm/kg. Baroreceptors sense changes in blood pressure

caused by alterations in blood volume and are peripherally located in the walls of

the left atrium, carotid sinus, and aortic arch (56). These receptors can respond to

changes in blood volume of more than 10%. In response to decreases in blood

pressure or volume, AVP is released and causes arteriolar vasoconstriction and

renal free–water conservation. This leads to a decrease in blood osmolality and an

increase in blood pressure. Activation of the renal renin–angiotensin system can

also activate AVP release.

MENSTRUAL CYCLE PHYSIOLOGY

[3] In the normal menstrual cycle, orderly cyclic hormone production and

parallel proliferation of the uterine lining prepare for implantation of the

embryo. Disorders of the menstrual cycle and, likewise, disorders of

menstrual physiology, may lead to various pathologic states, including

infertility, recurrent miscarriage, and malignancy.

Normal Menstrual Cycle

The normal human menstrual cycle can be divided into two segments: the

ovarian cycle and the uterine cycle, based on the organ under examination.

The ovarian cycle may be further divided into follicular and luteal phases,

whereas the uterine cycle is divided into corresponding proliferative and

secretory phases (Fig. 7-9). The phases of the ovarian cycle are characterized

as follows:

1. Follicular phase—hormonal feedback promotes the orderly development

of a single dominant follicle, which should be mature at midcycle and

prepared for ovulation. The average length of the human follicular phase

ranges from 10 to 14 days, and variability in this length is responsible for

most variations in total cycle length.

2. Luteal phase—the time from ovulation to the onset of menses has an

average length of 14 days.

A normal menstrual cycle lasts from 21 to 35 days, with 2 to 6 days of flow

and an average blood loss of 20 to 60 mL. However, studies of large numbers

of women with normal menstrual cycles showed that approximately twothirds of adult women have cycles lasting 21 to 35 days (57). The extremes of

299reproductive life (after menarche and perimenopause) are characterized by a

higher percentage of anovulatory or irregularly timed cycles (58,59).

Hormonal Variations

The relative pattern of ovarian, uterine, and hormonal variation along the

normal menstrual cycle is shown in Figure 7-9.

1. At the beginning of each monthly menstrual cycle, levels of gonadal

steroids are low and have been decreasing since the end of the luteal phase

of the previous cycle.

2. With the demise of the corpus luteum, FSH levels begin to rise, and a

cohort of growing follicles is recruited. These follicles each secrete

increasing levels of estrogen as they grow in the follicular phase. The

increase in estrogen is the stimulus for uterine endometrial proliferation.

3. Rising estrogen levels provide negative feedback on pituitary FSH

secretion, which begins to wane by the midpoint of the follicular phase. In

addition, the growing follicles produce inhibin B, which suppresses FSH

secretion by the pituitary. Conversely, LH initially decreases in response

to rising estradiol levels, but late in the follicular phase the LH level is

increased dramatically (biphasic response).

4. At the end of the follicular phase (just before ovulation), FSH-induced LH

receptors are present on granulosa cells and, with LH stimulation,

modulate the secretion of progesterone. Progesterone secretion is

responsible for the FSH midcycle surge.

5. After a sufficient degree of estrogenic stimulation, the pituitary LH surge

is triggered, which is the proximate cause of ovulation that occurs 24 to 36

hours later. Ovulation heralds the transition to the luteal–secretory phase.

6. The estrogen level decreases through the early luteal phase from just

before ovulation until the midluteal phase, when it begins to rise again as

a result of corpus luteum secretion. Similarly, inhibin A is secreted by the

corpus luteum.

7. Progesterone levels rise precipitously after ovulation and can be used as a

presumptive sign that ovulation has occurred.

8. Progesterone, estrogen, and inhibin A act centrally to suppress

gonadotropin secretion and new follicular growth. These hormones

remain elevated through the lifespan of the corpus luteum and wane with

its demise, thereby setting the stage for the next cycle.

300FIGURE 7-9 The menstrual cycle. The top panel shows the cyclic changes of folliclestimulating hormone (FSH), luteinizing hormone (LH), estradiol (E2), and progesterone (P)

relative to the time of ovulation. The bottom panel correlates the ovarian cycle in the

follicular and luteal phases and the endometrial cycle in the proliferative and secretory

phases.

Uterus

Cyclic Changes of the Endometrium

In 1950, Noyes, Hertig, and Rock described the cyclic histologic changes in the

301adult human endometrium (Fig. 7-10) (60). These changes proceed in an orderly

fashion in response to cyclic hormonal production by the ovaries (Fig. 7-9).

Histologic cycling of the endometrium can best be viewed in two parts: the

endometrial glands and the surrounding stroma. The superficial two-thirds of

the endometrium is the zone that proliferates and is ultimately shed with

each cycle if pregnancy does not occur. This cycling portion of the

endometrium is known as the decidua functionalis and is composed of a

deeply situated intermediate zone (stratum spongiosum) and a superficial

compact zone (stratum compactum). The decidua basalis is the deepest

region of the endometrium. It does not undergo significant monthly

proliferation but, instead, is the source of endometrial regeneration after

each menses (61).

302FIGURE 7-10 The number of oocytes in the ovary before and after birth and through

menopause.

The existence of endometrial stem cells was assumed but difficult to document.

Researchers found a small population of human epithelial and stromal cells that

possess clonogenicity, suggesting that they represent the putative endometrial

stem cells (62). Further evidence of the existence of such cells, and their source,

was provided by another study that showed endometrial glandular epithelial cells,

obtained from endometrial biopsies of women undergoing bone marrow

transplants, express the HLA type of the donor bone marrow (63). This finding

suggests that endometrial stem cells exist, reside in bone marrow, and migrate to

the basalis of the endometrium. Furthermore, the timing of the appearance of

these cells following the transplant was as long as several years. This experiment

has been duplicated using autologous bone marrow–derived stem cells and

placing them in the spiral arterioles of patients with intrauterine synechiae (64).

Animal models suggest this approach may be of value in regenerating damaged or

absent endometrium (65,66). It is likely that this treatment will prove to be of

clinical importance in patients with difficult to treat Asherman syndrome.

Proliferative Phase

[4] By convention, the first day of vaginal bleeding is called day 1 of the

menstrual cycle. After menses, the decidua basalis is composed of primordial

glands and dense scant stroma in its location adjacent to the myometrium.

The proliferative phase is characterized by progressive mitotic growth of the

decidua functionalis in preparation for implantation of the embryo in

response to rising circulating levels of estrogen (67). At the beginning of the

proliferative phase, the endometrium is relatively thin (1 to 2 mm). The

predominant change seen during this time is evolution of the initially

straight, narrow, and short endometrial glands into longer, tortuous

structures (68). Histologically, these proliferating glands have multiple

mitotic cells, and their organization changes from a low columnar pattern in

the early proliferative period to a pseudostratified pattern before ovulation.

Throughout this time, the stroma is a dense compact layer, and vascular

structures are infrequently seen.

Secretory Phase

In the typical 28-day cycle, ovulation occurs on cycle day 14. Within 48 to 72

hours following ovulation, the onset of progesterone secretion produces a

shift in histologic appearance of the endometrium to the secretory phase, so

named for the clear presence of eosinophilic protein-rich secretory products

303in the glandular lumen. In contrast to the proliferative phase, the secretory

phase of the menstrual cycle is characterized by the cellular effects of

progesterone in addition to estrogen. In general, progesterone’s effects are

antagonistic to those of estrogen, and there is a progressive decrease in the

endometrial cell’s estrogen receptor concentration. As a result, during the

latter half of the cycle, estrogen-induced DNA synthesis and cellular mitosis

are antagonized (67).

During the secretory phase, the endometrial glands form characteristic

periodic acid–Schiff positive–staining, glycogen-containing vacuoles. These

vacuoles initially appear subnuclearly and progress toward the glandular

lumen (Fig. 7-10) (60). The nuclei can be seen in the midportion of the cells

and ultimately undergo apocrine secretion into the glandular lumen, often by

cycle day 19 or 20. At postovulatory day 6 or 7, secretory activity of the

glands is generally maximal, and the endometrium is optimally prepared for

implantation of the blastocyst.

The stroma of the secretory phase remains unchanged histologically until

approximately the 7th postovulatory day, when there is a progressive

increase in edema. Coincident with maximal stromal edema in the late

secretory phase, the spiral arteries become clearly visible and progressively

lengthen and coil during the remainder of the secretory phase. By around

day 24, an eosinophilic-staining pattern, known as cuffing, is visible in the

perivascular stroma. Eosinophilia progresses to form islands in the stroma

followed by areas of confluence. This staining pattern of the edematous

stroma is termed pseudodecidual because of its similarity to the pattern that

occurs in pregnancy. Approximately 2 days before menses, there is a

dramatic increase in the number of polymorphonuclear lymphocytes that

migrate from the vascular system. This leukocytic infiltration heralds the

collapse of the endometrial stroma and the onset of the menstrual flow.

Menses

In the absence of implantation, glandular secretion ceases and an irregular

breakdown of the decidua functionalis occurs. The resultant shedding of this

layer of the endometrium is termed menses. The destruction of the corpus

luteum and its production of estrogen and progesterone is the presumed

cause of the shedding. With withdrawal of sex steroids, there is a profound

spiral artery vascular spasm that ultimately leads to endometrial ischemia.

Simultaneously, there is a breakdown of lysosomes and a release of

proteolytic enzymes, which further promote local tissue destruction. This

layer of endometrium is shed, leaving the decidua basalis as the source of

subsequent endometrial growth. Prostaglandins are produced throughout

304the menstrual cycle and are at their highest concentration during menses

(66). Prostaglandin F2α (PGF2α) is a potent vasoconstrictor, causing further

arteriolar vasospasm and endometrial ischemia. PGF2α produces

myometrial contractions that decrease local uterine wall blood flow and may

serve to expel physically the sloughing endometrial tissue from the uterus.

Dating the Endometrium

The changes seen in secretory endometrium relative to the LH surge were thought

to allow the assessment of the “normalcy” of endometrial development. Since

1950, it was felt that by knowing when a patient ovulated, it was possible to

obtain a sample of endometrium by endometrial biopsy and determine whether

the state of the endometrium corresponds to the appropriate time of the cycle.

Traditional thinking held that any discrepancy of more than 2 days between

chronologic and histologic date indicated a pathologic condition termed luteal

phase defect; this abnormality was linked to infertility (via implantation failure)

and early pregnancy loss (69).

Evidence suggests a lack of utility for the endometrial biopsy as a

diagnostic test for either infertility or early pregnancy loss (59). In a

randomized, observational study of regularly cycling, fertile women, it was found

that endometrial dating by hematoxylin and eosin staining is far less accurate and

precise than originally claimed and does not provide a valid method for the

diagnosis of luteal phase defect (70). Furthermore, a large prospective,

multicenter trial sponsored by the National Institutes of Health showed that

histologic dating of the endometrium does not discriminate between fertile and

infertile women (71). Thus, after half a century of using this test in the evaluation

of the subfertile couple, it became clear that the traditional endometrial biopsy has

no role in the routine evaluation of infertility or early pregnancy loss.

Given the lack of histologic efficacy in evaluating the receptivity of the

endometrium, investigation turned to the use of molecular and genetic markers.

Cyclin E and p27 were found to be credible markers to discern endometrial

receptivity (72,73). Microarray technology has been utilized to link gene

expression to functionally receptive endometrium, with promising results (74,75).

Ovarian Follicular Development

The number of oocytes peaks in the fetus at 6 to 7 million by 20 weeks of

gestation (Fig. 7-10) (76). Simultaneously (and peaking at the 5th month of

gestation), atresia of the oogonia occurs, rapidly followed by follicular atresia. At

birth, only 1 to 2 million oocytes remain in the ovaries, and at puberty, only

300,000 of the original 6 to 7 million oocytes are available for ovulation

305(76,77). Of these, only 400 to 500 will ultimately be released during ovulation.

By the time of menopause, the ovary will be composed primarily of dense stromal

tissue with only rare interspersed oocytes remaining.

A central dogma of reproductive biology is that in postnatal mammalian

females there is no capacity for oocyte production. Because oocytes enter the

diplotene resting stage of meiosis in the fetus and persist in this stage until

ovulation, much of the DNA, proteins, and messenger RNA (mRNA) necessary

for development of the preimplantation embryo is synthesized by this stage. At

the diplotene stage, a single layer of 8 to 10 granulosa cells surrounds the oogonia

to form the primordial follicle. The oogonia that fail to become properly

surrounded by granulosa cells undergo atresia (78). The remainder proceeds with

follicular development. Thus, most oocytes are lost during fetal development, and

the remaining follicles are steadily “used up” throughout the intervening years

until menopause.

Evidence has begun to challenge this theory. Studies in the mouse showed that

production of oocytes and corresponding folliculogenesis can occur well into

adult life (79). The reservoir of germline stem cells responsible for this oocyte

development appears to reside in the bone marrow (80). While stem cells have

been found in the human adult ovary (81,82), it is not clear if these cells are true

ovarian germline stem cells and if they play a physiologic role within the ovary

regarding follicular development (82,83).

Meiotic Arrest of Oocyte and Resumption

Meiosis (the germ cell process of reduction division) is divided into four

phases: prophase, metaphase, anaphase, and telophase. The prophase of

meiosis I is further divided into five stages: leptotene, zygotene, pachytene,

diplotene, and diakinesis.

Oogonia differ from spermatogonia in that only one final daughter cell

(oocyte) forms from each precursor cell, with the excess genetic material

discarded in two polar bodies. When the developing oogonia begin to enter

meiotic prophase I, they are known as primary oocytes (84). This process

begins at roughly 8 weeks of gestation. Only those oogonia that enter meiosis will

survive the wave of atresia that sweeps the fetal ovary before birth. The oocytes

arrested in prophase (in the late diplotene or “dictyate” stage) will remain thus

until the time of ovulation, when the process of meiosis resumes. The mechanism

for this mitotic stasis is believed to be an oocyte maturation inhibitor (OMI)

produced by granulosa cells (85). Granulosa-derived cAMP seems to be

implicated in inhibiting germinal vesicle breakdown and meiosis resumption (86).

This inhibitor gains access to the oocyte via gap junctions connecting the oocyte

and its surrounding cumulus of granulosa. These intercellular channels are formed

306by proteins known as connexins. With the midcycle LH surge, the gap junctions

are disrupted, granulosa cells are no longer connected to the oocyte, and meiosis I

is allowed to resume.

Follicular Development

Follicular development, also known as folliculogenesis, is a dynamic process

that continues from menarche until menopause. The process is designed to

allow the monthly recruitment of a cohort of primordial follicles and,

ultimately, to release a single, mature, dominant follicle during ovulation

each month. Therefore, it is highly coordinated with oocyte maturation.

Folliculogenesis has been divided into different steps according to follicular

characteristics regarding the number and appearance of granulosa cells,

development of theca cells and formation of a fluid-filled structure known as

antrum. Preantral follicles include primordial, primary, and secondary follicles.

Antral follicles include tertiary and preovulatory follicles.

Primordial follicles are 0.03 to 0.05 mm in diameter structures formed by a

primary oocyte (arrested in prophase of meiosis I), surrounded by one layer of

flattened granulosa cells contained by the basal lamina.

Primary follicles are 0.1 mm follicles formed when granulosa cells are still a

one cell layer but acquire a cuboidal form. This is the first sign of follicular

recruitment. Protein synthesis and secretion form an extracellular matrix capsule

known as the zona pellucida, traversed by intercellular channels (gap unions) that

maintain active connections between granulosa cells and the oocyte. Granulosa

cells in the primary follicle develop FSH receptors, without endocrine effect as a

result of the absence of follicular vascularization and, therefore, nonexistent

exposure to circulating FSH.

Secondary follicles are 0.2 mm in size and develop several layers of cuboidal

granulosa cells with marked expression of FSH receptors. Stromal cell in contact

with the granulosa and basal lamina are differentiated into theca cells with LH

receptor expression. In the theca layer neoangiogenesis occurs, vascularizing the

follicle and exposing it to circulating FSH and LH.

Tertiary follicles are characterized by the formation of the antral cavity or

antrum, as a consequence of granulosa cell secretion intercellular accumulation.

Early tertiary follicles are 0.2 to 5 mm in size and at this point the theca layer is

divided into theca interna and theca externa, which forms a transition with the

ovarian stroma. Late tertiary follicles are 10 to 20 mm in size. Their large antral

cavity divides granulosa in several cell populations, the corona radiata in contact

with the oocyte, mural (membranous) granulosa in contact with the follicular wall

and the cumulus ophorus that appears as a stalk joining the corona radiata and the

mural granulosa.

307Preovulatory follicles are the final stage of follicular development and >20

mm in size, structures from which ovulation occurs. Late in this stage and before

ovulation, the primary oocyte completes meiosis I, becoming a secondary oocyte

arrested in metaphase of meiosis II. Late tertiary/preovulatory follicles are also

known as Graafian follicles.

Gonadotropin dependence in folliculogenesis is conditioned by the expression

of FSH and LH receptors in granulosa and theca cells, respectively, and by the

presence of follicular vascularization. Considerable expression of granulosa FSH

receptors and formation of vascularized theca layer occurs in the secondary

follicle. Consequently, follicular development is gonadotropin independent up to

the formation of secondary follicles or late preantral phase. Early antral follicle

development and its maturation process up to a preovulatory follicle is a

gonadotropin dependent phase.

Primordial Follicles

The initial recruitment and growth of the primordial follicles is gonadotropin

independent and affects a cohort over several months (87). The stimuli

responsible for the recruitment of a specific cohort of follicles in each cycle are

yet to be understood, but it seems to be under autocrine and paracrine control.

Interaction between oocyte and neighboring granulosa cells seems to be

fundamental for oocyte growth development, granulosa cell proliferation and the

resultant primordial follicle activation.

Maintenance of a population of dormant primordial follicles is the basis for

guaranteeing an oocyte supply throughout reproductive life (88). Whether

secretion of stimulating or inhibiting factors is involved in recruitment regulation

is being studied, although accelerated recruitment in isolated primordial follicles

cultured in vitro suggests inhibitory mechanisms can have a more important role

(89). Several factors have been implicated with an inhibitory effect over

primordial follicle activation, such as anti-mullerian hormone (AMH) (90),

phosphate and tensin homolog (PTEN) (91), tuberin/tuberous sclerosis complex

(TSC) (92), Forkhead boxL2 (Foxl2) (93), and Forkhead box O3 (FOXO3a) (94).

Their expression is responsible for preservation of primordial follicular dormancy

and depletion of these factors in knockout mice has been associated with

premature activation and early depletion of primordial follicles. On the other

hand, phosphotidylinositol-3-kinase signaling mediated by 3-phosphoinositide

dependent kinase-1 (PDK1), and mammalian target of rapamycin complex-1

(mTORC1), and S6 kinase-ribosomal protein (S6K1-rpS6), have been related to

primordial follicle activation and survival (95–98).

Preantral Follicle

308At the secondary follicle stage, after initial recruitment, FSH assumes control of

follicular differentiation and growth and allows a cohort of follicles to continue

differentiation. This process signals the shift from gonadotropin-independent to

gonadotropin-dependent growth. The decline in luteal phase estrogen,

progesterone, and inhibin A production by the now fading corpus luteum from the

previous cycle allows the increase in FSH that stimulates this follicular growth

(99).

Simultaneously, theca cells in the stroma bordering the granulosa cells

proliferate. Both cell types function synergistically to produce estrogens that are

secreted into the systemic circulation. At this stage of development, each of the

seemingly identical cohort members must be either selected for dominance or

undergo atresia. It is likely that the follicle destined to ovulate was selected before

this point, although the mechanism for selection remains obscure.

Two-Cell, Two-Gonadotropin Theory

The fundamental tenet of follicular development is the two-cell, twogonadotropin theory (Fig. 7-11) (87,100,101). This theory states that there is

a subdivision and compartmentalization of steroid hormone synthesis

activity in the developing follicle. Most aromatase activity (for estrogen

production) is in the granulosa cells (102). Aromatase activity is enhanced by

FSH stimulation of specific receptors on these cells (103,104). Granulosa cells

lack several enzymes that occur earlier in the steroidogenic pathway and require

androgens as a substrate for aromatization. Androgens, in turn, are synthesized

primarily in response to stimulation by LH, and the theca cells possess most of

the LH receptors at this stage (103,104). Therefore, a synergistic relationship

must exist: LH stimulates the theca cells to produce androgens (primarily

androstenedione), which are transferred to the granulosa cells for FSH-stimulated

aromatization into estrogens. These locally produced estrogens create a

microenvironment within the follicle that is favorable for continued growth and

nutrition (105). FSH and local estrogens serve to further stimulate estrogen

production, FSH receptor synthesis and expression, and granulosa cell

proliferation and differentiation.

Androgens have two positive regulatory roles in follicular development.

Within the ovary, androgens promote granulose cell proliferation, aromatase

activity, and inhibit programmed death of these cells (106).

As the peripheral estrogen level rises, it negatively feeds back on the

pituitary and hypothalamus to decrease circulating FSH levels (107).

Increased ovarian production of inhibin B further decreases FSH production

at this point.

The falling FSH level that occurs with the progression of the follicular

309phase represents a threat to continued follicular growth. The resulting adverse

environment can be withstood only by follicles with a selective advantage for

binding the diminishing FSH molecules; that is, those with the greatest number of

FSH receptors. The dominant follicle, therefore, can be perceived as the one with

a richly estrogenic microenvironment and the most FSH receptors (108). Increase

in FSH receptors results from an increase in granulosa cell population, because

FSH receptor number is similar and constant in each granulosa cell (109,110). As

it grows and develops, the follicle continues to produce estrogen, which results in

further lowering of the circulating FSH and creates a more adverse environment

for competing follicles. This process continues until all members of the initial

cohort, with the exception of the single dominant follicle, have suffered atresia.

The stage is set for ovulation.

Chronic elevation of androgens suppresses hypothalamic–pituitary secretion of

FSH, a detriment to the development and maturation of a dominant follicle (106).

Clinically, androgen excess results in chronic anovulation, as is seen in polycystic

ovarian syndrome.

FIGURE 7-11 The two-cell, two-gonadotropin theory of follicular development in which

there is compartmentalization of steroid hormone synthesis in the developing follicle. LH,

luteinizing hormone; FSH, follicle-stimulating hormone.

Preovulatory Follicle

Preovulatory follicles are characterized by a fluid-filled antrum that is

311composed of plasma with granulosa cell secretions. The granulosa cells at this

point have further differentiated into a heterogeneous population. The oocyte

remains connected to the follicle by a stalk of specialized granulosa known as the

cumulus oophorus.

Rising estrogen levels have a negative feedback effect on FSH secretion.

Conversely, LH undergoes biphasic regulation by circulating estrogens. At

lower concentrations, estrogens inhibit LH secretion. At higher levels,

estrogen enhances LH release. This stimulation requires a sustained high level

of estrogen (>200 pg/mL) for more than 48 hours (111). When the rising estrogen

level produces positive feedback, a substantial surge in LH secretion occurs.

Concomitant to these events, the local estrogen–FSH interactions in the

dominant follicle induce LH receptors on the granulosa cells. Exposure to high

levels of LH results in a specific response by the dominant follicle—the result is

luteinization of the granulosa cells, production of progesterone, and initiation of

ovulation. Late follicular phase progesterone secretion is responsible for the FSH

midcycle surge that stimulates plasminogen activator, LH granulosa cell receptor

formation, and debilitates oocyte binding to the follicular wall (110). Ovulation

will occur in the single mature, or Graafian, follicle 10 to 12 hours after the LH

peak or 34 to 36 hours after the initial rise in midcycle LH (112–114).

The sex steroids are not the only gonadotropin regulators of follicular

development. Two related granulosa cell–derived peptides were identified that

play opposing roles in pituitary feedback (115). The first of these peptides,

inhibin, is secreted in two forms: inhibin A and inhibin B. Inhibin B is

secreted primarily in the follicular phase and is stimulated by FSH, whereas

inhibin A is mainly active in the luteal phase (116). Both forms of inhibin act to

inhibit FSH synthesis and release (117,118). The second peptide, activin,

stimulates FSH release from the pituitary gland and potentiates its action in the

ovary (119,120). It is likely that there are numerous other intraovarian regulators

similar to inhibin and activin, each of which may play a key role in promoting the

normal ovulatory process (121). Some of these include follistatin, insulin-like

growth factor-1 (ILGF-1), (EGF)/transforming growth factor-α (TGF-α), TGF-β1,

growth differentiation factor 9 (GDF-9) (122,123), fibroblast growth factor-β

(FGF-β), interleukin-1, tissue necrosis factor-α, OMI, and renin–angiotensin.

Anti-mullerian hormone, produced exclusively by granulosa cells of growing

primary and preantral follicles, is the most accurate reflection of ovarian reserve

and seems to influence the dominant follicle selection by decreasing FSH

sensitivity at receptor level, thus inhibiting the initial selection of preantral and

small antral follicles (124–126).

Ovulation

312The midcycle LH surge is responsible for a dramatic increase in local

concentrations of prostaglandins and proteolytic enzymes in the follicular

wall (127). These substances progressively weaken the follicular wall, allowing

the formation of a bleb-like superficial follicular protrusion known as the stigma

and ultimately the wall’s perforation. Ovulation most likely represents a slow

extrusion of the oocyte through this opening in the follicle rather than a rupture of

the follicular structure (128). Direct measurements of intrafollicular pressures

were recorded and failed to demonstrate an explosive event.

Luteal Phase

Structure of Corpus Luteum

After ovulation, the remaining follicular shell is transformed into the

primary regulator of the luteal phase: the corpus luteum. Membranous

granulosa cells remaining in the follicle begin to take up lipids and the

characteristic yellow lutein pigment for which the structure is named. These cells

are active secretory structures that produce progesterone, which supports the

endometrium of the luteal phase. In addition, estrogen and inhibin A are produced

in significant quantities. Unlike the process that occurs in the developing follicle,

the basement membrane of the corpus luteum degenerates to allow proliferating

blood vessels to invade the granulosa-luteal cells in response to secretion of

angiogenic factors such as vascular endothelial growth factor (129). This

angiogenic response allows large amounts of luteal hormones to enter the

systemic circulation.

Hormonal Function and Regulation

The hormonal changes of the luteal phase are characterized by a series of

negative feedback interactions designed to lead to regression of the corpus

luteum if pregnancy does not occur. Corpus luteum steroids (estradiol and

progesterone) provide negative central feedback and cause a decrease in FSH

and LH secretion. Continued secretion of both steroids will decrease the

stimuli for subsequent follicular recruitment. Similarly, luteal secretion of

inhibin potentiates FSH withdrawal. In the ovary, local production of

progesterone inhibits the further development and recruitment of additional

follicles.

Continued corpus luteum function depends on continued LH production.

In the absence of this stimulation, the corpus luteum will invariably regress after

12 to 16 days and form the scar-like corpora albicans (130). The exact

mechanism of luteolysis is unclear and most likely involves local paracrine

factors. In the absence of pregnancy, the corpus luteum regresses, and estrogen

and progesterone levels wane. This removes central inhibition on gonadotropin

313secretion and allows FSH and LH levels to rise and recruit another cohort of

follicles.

If pregnancy does occur, placental hCG will mimic LH action and

continually stimulate the corpus luteum to secrete progesterone. Successful

implantation results in hormonal support to allow continued maintenance of the

corpus luteum and the endometrium. Evidence from patients undergoing oocyte

donation cycles demonstrated that continued luteal function is essential for

continuation of the pregnancy until approximately 5 weeks of gestation, when

sufficient progesterone is produced by the developing placenta (131). This switch

in the source of regulatory progesterone production is referred to as the luteal–

placental shift.

Summary of Menstrual Cycle Regulation

Following is a summary of the regulation of the menstrual cycle:

1. GnRH is produced in the arcuate nucleus of the hypothalamus and

secreted in a pulsatile fashion into the portal circulation, where it travels

to the anterior pituitary.

2. Ovarian follicular development moves from a period of gonadotropin

independence to a phase of FSH dependence.

3. As the corpus luteum of the previous cycle fades, luteal production of

progesterone and inhibin A decreases, allowing FSH levels to rise.

4. In response to FSH stimulus, the follicles grow, differentiate, and secrete

increasing amounts of estrogen and inhibin B.

5. Estrogen stimulates growth and differentiation of the functional layer of

the endometrium, which prepares for implantation. Estrogens work with

FSH in stimulating follicular development.

6. The two-cell, two-gonadotropin theory dictates that with LH stimulation,

the ovarian theca cells will produce androgens that are converted by the

granulosa cells into estrogens under the stimulus of FSH.

7. Rising estrogen and inhibin levels negatively feedback on the pituitary

gland and hypothalamus and decrease the secretion of FSH.

8. The one follicle destined to ovulate each cycle is called the dominant

follicle. It has relatively more FSH receptors and produces a larger

concentration of estrogens than the follicles that will undergo atresia. It is

able to continue to grow despite falling FSH levels.

9. Sustained high estrogen levels cause a surge in pituitary LH secretion that

triggers ovulation, progesterone production, and the shift to the secretory,

or luteal, phase.

10. Luteal function is dependent on the presence of LH. The corpus luteum

314secretes estrogen, progesterone, and inhibin A, which serve to maintain

gonadotropin suppression. Without continued LH secretion, the corpus

luteum will regress after 12 to 16 days. The resulting loss of progesterone

secretion results in menstruation.

11. If pregnancy occurs, the embryo secretes hCG, which mimics the action of LH

by sustaining the corpus luteum. The corpus luteum continues to secrete

progesterone and supports the secretory endometrium, allowing the pregnancy

to continue to develop.

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