Berek Novak's Gyn 2019. Chapter 22 Primary Care

 CHAPTER 22

Primary Care

KEY POINTS

1 Respiratory infections in adults are commonly viral and do not require antibiotics.

For good antibiotic stewardship, one needs to use them only for bacterial infections

that require them. If empiric therapy is used, it should be based on the specific

patient and the severity of the infection. All patients with possible communityacquired pneumonia should have a chest radiograph to establish the diagnosis and

presence of complications.

2 Effective screening for hypertension and hyperlipidemia is critical to reduce the

occurrence of cardiac disease (a primary cause of death). When hypertension or

significant risks for hypertension are found, active lifestyle intervention needs to be

initiated. If this is not adequate, pharmaceutical intervention is used to achieve a

goal of less than 140/90. In patients with comorbidities such as diabetes or renal

disease, the goal should be less than 130/80.

3 The role of diet in hyperlipidemia is still unclear although a low-fat diet along with

weight loss and exercise do reduce lipids. Current recommendations strongly

encourage the use of statins as first line pharmaceutical therapy with clear guidelines

for use and optimal goals as targets.

11474 Type 2 diabetes is increasing as the incidence of obesity increases. Screening highrisk individuals allows early diagnosis and intervention prior to development of

complications. Lifestyle modifications including diet, weight loss, and exercise are

the first steps in management.

5 Given the frequency of thyroid pathology in women, providers need to understand

risk factors that merit screening and the proper physical examination to identify

masses. The sensitive thyroid-stimulating hormone (TSH) assay is the single best

screening test for hyperthyroidism and hypothyroidism.

As health care providers for women, gynecologists are responsible for providing

care that extends beyond diseases of the reproductive organs to include much of

the general medical care of their patients. Broadening the spectrum of care

requires adjustments in practice, with less emphasis placed on the surgical aspects

of the specialty. Early diagnosis and treatment of medical illnesses can have a

major impact on a woman’s health. Although timely referral is important for

complex and advanced diseases, many conditions can be screened for,

recognized, and potentially treated initially by gynecologists.

Respiratory problems are the most common reasons patients seek care

from a physician, so gynecologists should be aware of their pathophysiology.

Cardiovascular disease has a significant impact on the overall morbidity and

is the main cause of death in women. Cardiovascular disease is associated

with cigarette smoking, hypertension, hypercholesterolemia, and diabetes

mellitus (DM). These conditions are responsive to screening, behavior

modification, and control to lower risk factors. Thyroid disease is a major

cause of morbidity for women. Because of the interaction of hormones and

the overall effect on the endocrine system, thyroid disease can be of special

significance in women. The gynecologist should provide screening and initial

therapy for these conditions and assess the need for referral.

RESPIRATORY INFECTIONS

Infections of the respiratory system can range from the common cold to lifethreatening illness. Those with risk factors should be counseled about preventive

measures. Vaccines against flu and pneumonia should be offered as indicated.

Upper Respiratory Infections (URIs)

This term can encompass a number of diagnoses including the “common cold.”

“Cold” is a term often used for a variety of virus-induced mild URIs that typically

have the symptoms of stuffy nose, sore scratchy throat, cough, no or low-grade

fever, and fatigue or malaise (1). Ear pain can be part of the cluster. Despite

1148thoughts that “colds” are more common in certain times of the year, there is no

seasonal variation in their incidence—only in the virus causing the cold.

Adenovirus, rhinoviruses, coronaviruses, and respiratory syncytial viruses are

common etiologies of “colds.” Although patients will frequently equate colds and

“flu,” the viruses that cause influenza tend to have more body aches, fever, and

systemic symptoms as well as being seasonal.

Differentiating which virus is causing a cold does not impact treatment, so

cultures are not indicated unless there is concern for an influenza virus that might

benefit from antiviral medication. The diagnosis of a cold tends to be a process of

exclusion. The presence of temperature >100, facial pain, prolonged (>2 weeks)

barking cough, exudate on pharynx/tonsils, abnormal breath sounds, or poor

oxygen saturation would indicate that other diagnoses need to be considered, such

as sinusitis, pertussis, strep throat, bronchitis, monospot, or influenza. In the

presence of these findings, strep culture, pertussis screen, viral screen for

influenza, or chest x-ray might be indicated.

The treatment of a cold is basically symptomatic. This includes aspirin/NSAID

for any body aches or low-grade temperature, hydration, decongestant (topical or

oral), and good hand hygiene. In an otherwise healthy person a cold will last 7 to

10 days and occasionally up to 2 weeks. Spread is by droplets (both small from

cough/sneeze and large on hands/environmental) and contact (hands or

contaminated surfaces). Antibacterial wipes and cleaners do NOT impact the

transmission of cold viruses (2). The use of decongestants such as

pseudoephedrine or oxymetazoline HCl should not be used for more than 2 or 3

days because of a risk of a rebound effect.

The risk of acquiring a cold is increased in individuals who are sleep deprived,

stressed, have children in day care settings, have chronic diseases, smoke, or have

poor nutrition and immune deficiency. The last four situations increase the risk of

a more severe “cold” and having it progress into a bacterial complication.

Seasonal changes do NOT change the incidence of “colds” but only the virus that

caused it.

Sinusitis

A problem frequently encountered in women is self-diagnosed “sinus

problems.” Many medical problems—headaches, dental pain, postnasal drainage,

halitosis, and dyspepsia—may be related to sinus conditions. The sinuses are not

an isolated organ, and diseases of the sinuses are often related to conditions that

affect other portions of the respiratory system (i.e., the nose, bronchial tree, and

lungs). Therefore, during the evaluation of symptoms attributable to sinusitis, the

presence of other infections should be investigated.

Multiple infectious and chemical agents or reactions to nervous, physical,

1149emotional, or hormonal stimuli may cause an inflammatory response in the

respiratory system (3). Systemic diseases such as connective tissue syndromes

and malnutrition may contribute to chronic sinusitis. Environmental factors in the

workplace and geographic conditions (e.g., cold and damp weather) may

aggravate or accelerate the development of sinusitis. Factors contributing to the

development of sinus disease include atmospheric pollutants, allergy, tobacco

smoke, skeletal deformities, dental conditions, barotrauma from scuba diving or

airline travel, and neoplasms.

[1] Most acute infections (lasting less than 4 weeks) begin with a viral agent

(acute viral rhinosinusitis [AVRS]) in the nose or nasopharynx that causes

inflammation, blocking the draining ostia (3). The location of the symptoms

varies by the anatomic site of infection—maxillary sinus over the cheeks, ethmoid

sinus across the nose, frontal sinus in the supraorbital area, and sphenoid sinus to

the vertex of the head—and typically last 7 to 10 days, clearing with nothing

more than a decongestant. Viral agents impede the sweeping motion of ciliary

function in the sinus and, in combination with edema from inflammation,

may occasionally lead to superinfection with bacteria (acute bacterial

rhinosinusitis [ABRS]). The most common bacterial agents infecting sinuses

are Streptococcus pneumoniae and Haemophilus influenzae. Gram-negative

organisms are usually limited to compromised hosts in intensive care units. [1]

Although less than 2% of acute sinusitis cases transition from viral to bacterial

infections requiring antibiotics, more than 85% of patients receive antibiotic

prescriptions. Chronic sinusitis (lasting more than 12 weeks) develops from either

inadequate drainage or compromised local defense mechanisms. The flora usually

is polymicrobial, consisting of aerobic and anaerobic organisms.

Sinus ailments frequently occur in middle-age individuals. Acute infection

is usually located in the maxillary and frontal sinuses. Classically, infection in the

maxillary sinus results from obstruction of the ostia found in the medial wall of

the nose. Fever, malaise, a vague headache, and pain in the maxillary teeth are

early symptoms. Reports of “fullness” in the face or exploding pressure behind

the eyes often are elicited as well as increasing pain with bending over. Pressure

and percussion over the malar areas can cause severe pain. Purulent exudates in

the middle meatus of the nose or in the nasopharynx often are present. To

differentiate between a “cold” and sinusitis the following can be helpful. Viral

URI typically peak rapidly in 3 to 4 days and they consistently decline in severity

of symptoms with full resolution in 7 to 14 days. Sinusitis in contrast will often

persistent without improvement for over a week. A pattern of initial improvement

with sudden worsening may represent a transition to a bacterial infection. Initial

episodes of sinusitis do not require imaging studies; however, when persistent

infections occur, studies and referral are indicated. Radiographic changes do not

1150reliably identify sinusitis secondary to bacteria. Unless culture samples are

obtained by direct needle drainage, they are contaminated by oropharyngeal flora

and are thus of no value. For this reason, therapy usually is empiric.

Systemic decongestants containing pseudoephedrine are useful in shrinking

the obstructive ostia and promoting sinus drainage and ventilation. Topical

decongestants should be used for no longer than 3 days because prolonged use

may lead to rebound vasodilation and worsening of symptoms. Mucolytics like

guaifenesin may help thin sinus secretions and promote drainage. Antihistamines

should be avoided in acute sinusitis because of their drying effects, which can

lead to thickened secretions and poor drainage of the sinuses. Analgesics are

recommended for pain relief. Therapies to relieve symptoms include facial hot

packs and analgesics. Topical nasal steroids may accelerate the recovery in

patients with viral sinusitis and those with a history of chronic rhinitis or recurrent

sinusitis who seek treatment of acute rhinosinusitis (4,5). Improvement should be

apparent within 48 hours of treatment, but 10 days may be necessary for complete

resolution of symptoms. If antibiotics are used, broad antibiotic coverage of

common aerobes and anaerobes is necessary but should be limited to patients

with acute pain, especially unilateral maxillary tooth, facial, or sinus pain,

and purulent discharge, particularly if the symptoms initially improved and

then worsened. This cluster of symptoms is more suggestive of bacterial

rather than viral acute sinusitis. It should be noted that the majority of acute

bacterial sinusitis cases resolve in 7 to 10 days without antibiotics, similarly

to the viral form. [1] For this reason, in an otherwise healthy adult, the use of

antibiotics is not recommended. In the setting of comorbidities such as diabetes,

chronic respiratory disease, congestive failure or immunodeficiency state, the use

of antibiotics for ABRS may be warranted. For acute bacterial sinus infections,

amoxicillin (1,000 mg three times a day) remains the treatment of choice.

Amoxicillin is inexpensive, penetrates the sinus tissues well, and can be changed

to another antibiotic if symptoms have not improved in 48 to 72 hours. If these

give only a minimal or no response after 7 days, consider broader-spectrum

antibiotics. If beta-lactam resistance is likely, amoxicillin/clavulanic acid (875 mg

twice daily) may be used. Other second-line drugs include, levofloxacin (500 mg

qd), and doxycycline (200 mg qd for 5 to 10 days). The usual treatment course is

5 to 10 days, and patients should be informed that relapses might occur if the full

course of treatment is not completed. [1] Trimethoprim/sulfamethoxazole and

azithromycin are no longer recommended as a result of high rates of microbial

resistance (3).

No clinical criteria can reliably identify those patients who might benefit

from treatment with antibiotics. It is reasonable to treat women with presumed

bacterial sinusitis if they have high fever, systemic toxicity, immune deficiency,

1151or possible orbital or intracranial involvement (5). Although very rare, untreated

sinus infections may have dire consequences, such as orbital cellulitis, leading to

orbital abscess, subperiosteal abscess formation of the facial bones, cavernous

sinus thrombosis, and acute meningitis. Brain and dural abscesses are rare; when

they occur, it usually is the result of direct spread from a sinus. A patient

complaining of abnormal vision such as diplopia, changes in mental status, and

periorbital edema should prompt a referral to the emergency room for evaluation

of intracranial or orbital extension. Computed tomography scanning is the most

accurate diagnostic tool. The use of aggressive surgical approaches with broadspectrum antibiotics is necessary for adequate drainage.

Otitis Media

Otitis media remains primarily a disease of children, but may affect adults,

often secondary to a concurrent viral infection of the upper respiratory tract.

Diagnosis in most cases reveals fluid behind the tympanic membrane. Treatment

is directed to symptoms and involves the use of antihistamines and decongestants,

despite few data to support their use for acute serous otitis, as this is typically

caused by a blocked eustachian tube. Acute suppurative otitis media is usually a

bacterial infection; S. pneumoniae and H. influenzae are the most common

pathogens. [1] Symptoms include acute purulent otorrhea, fever, hearing loss,

severe deep throbbing ear pain, and leukocytosis. Physical examination of the ear

reveals a red, bulging, or perforated membrane with possible pre- and

postauricular nodes. Indicated treatment is broad-spectrum antibiotics such as

amoxicillin, amoxicillin/clavulanic acid, cefuroxime, erythromycin, or

azithromycin (6,7).

Bronchitis

Acute bronchitis is an inflammatory condition of the tracheobronchial tree.

Most often it is viral in origin and occurs in winter. It accounts for up to 10%

of ambulatory care visits. Common cold viruses (rhinovirus and coronavirus),

adenovirus, influenza virus, and Mycoplasma pneumoniae (a nonviral pathogen)

are the most common pathogens involved. Bacterial infections occur less

commonly and may be secondary pathogens. Cough, hoarseness, and mild fever

are the usual presenting symptoms. In the initial 3 to 4 days, the symptoms of

rhinitis and sore throat are prominent; coughing may last as long as 3 weeks.

Presence of tachycardia or tachypnea raises concern for pneumonia (8,9). The

prolonged nature of these infections promotes the use of antibiotics to “clear up

the infection” (8). Sputum production commonly occurs and may be prolonged in

cigarette smokers. [1] Most serious bacterial infections occur in cigarette

1152smokers, who have damage to the lining of the upper respiratory tree and changes

in the host flora. Differential diagnosis includes the following: postnasal drip,

asthma, pneumonia, gastroesophageal reflex disease (GERD), use of angiotensinconverting enzyme (ACE) inhibitors, and heart failure.

Physical examination discloses a variety of upper airway sounds, usually

coarse rhonchi. Rales are usually not present on auscultation, and signs of

consolidation and alveolar involvement are absent. During auscultation of the

chest, signs of pneumonia such as fine rales, decreased breath sounds, and

euphonia (“E to A changes”) should be sought. If the results of the physical

examination are uncertain or the patient’s condition appears to be in respiratory

distress chest radiography should be performed to detect the presence of

parenchymal disease. Paradoxically, as the initial acute syndrome subsides,

sputum production may become more purulent. Sputum cultures are of limited

value because of the polymicrobial nature of infections. In the absence of

complications, treatment is directed to relief of symptoms. [1] The use of

antibiotics is reserved for patients in whom chest radiography findings are

consistent with pneumonia (10,11). Cough is usually the most aggravating

symptom and may be treated with antitussive preparations containing either

dextromethorphan or guaifenesin. The use of codeine as a cough suppressant is

discouraged. The efficacy of any expectorant is not proved. If the cough persists

longer than 2 weeks the patient may have pertussis. This is treated with

azithromycin or other macrolides (8).

Chronic bronchitis is defined as a productive cough from excessive

secretions for at least 3 months in a year for 2 consecutive years. Prevalence is

estimated to be between 10% and 25% of the adult population who are smokers.

Previously the incidence was lower in women than men, but as the prevalence of

cigarette smoking in women increased, so too has the incidence of bronchitis in

women. Chronic bronchitis is classified as a form of chronic obstructive

pulmonary disease (COPD; e.g., “blue bloaters”). Other causes include chronic

infections and environmental pathogens found in dust. The cardinal manifestation

of disease is an incessant cough, usually in the morning, with expectoration of

sputum. Because of frequent exacerbations, the hospitalizations involved and the

complexity of medical management, these patients should be referred to an

internist.

Pneumonia

Pneumonia is defined as inflammation of the distal lung that includes

terminal airways, alveolar spaces, and the interstitium. Pneumonia may have

multiple causes, including viral and bacterial infections or aspiration. Aspiration

pneumonia is usually the result of depressed awareness commonly associated

1153with the use of drugs and alcohol or anesthesia. Viral pneumonias are caused by

multiple infectious agents, including influenza A or B, parainfluenza virus, or

respiratory syncytial virus. Most viral syndromes are spread by aerosolization

associated with coughing, sneezing, and even conversation. Incubation is short,

requiring only 1 to 3 days before the acute onset of fever, chills, headache,

fatigue, and myalgias. Symptom intensity is directly related to intensity of the

host febrile reaction. Pneumonia develops in only 1% of patients who have a viral

syndrome, but mortality rates may reach 30% in immunocompromised

individuals and the elderly. An additional risk is the development of secondary

bacterial pneumonias after the initial viral insult. These infections are more

common in elderly patients and may explain the high fatality in this group (12).

Staphylococcal pneumonias, which often arise from a previous viral infection, are

extremely lethal regardless of patient age. [1] The best treatment for viral

pneumonia is prevention by immunization. Treatment is supportive and consists

mostly of administration of antipyretics and fluids.

Bacterial pneumonia is classified as either community-acquired (CAP) or

nosocomial, and in many cases the classification determines prognosis and

antibiotic therapy. [1] Risk factors that contribute to mortality are chronic

cardiopulmonary diseases, alcoholism, diabetes, renal failure, malignancy, and

malnutrition. Prognostic features associated with poor outcome include greater

than two lobe involvement, respiratory rate greater than 30 breaths per minute on

presentation, severe hypoxemia (<60 mm Hg on room air), hypoalbuminemia,

and septicemia. Pneumonia is a common cause of adult respiratory distress

syndrome (ARDS), with a mortality rate between 50% and 70% (12,13). CAP is

the most common cause of severe sepsis and a leading cause of death from

infection in the United States.

Signs and symptoms of pneumonia vary depending on the infecting

organism and the patient’s immune status. In typical pneumonias, the usual

presentation is a patient with high fever, rigors, productive cough, chills, and

pleuritic chest pain. Chest radiography often will show infiltrates (11). The

following agents, listed in decreasing order, cause two-thirds of all bacterial

pneumonias: S. pneumoniae, H. influenzae, Klebsiella pneumoniae, gramnegative organisms, and anaerobic bacteria. Atypical pneumonias are more

insidious in onset than typical pneumonias. Patients have moderate fever without

the characteristic rigors and chills. Additional symptoms include a nonproductive

cough, headache, myalgias, and mild leukocytosis. Chest radiography reveals

bronchopneumonia with a diffuse interstitial pattern; characteristically, the patient

does not appear to be as ill as the x-ray suggests. Common causes of atypical

pneumonia include viruses, M. pneumoniae, Legionella pneumophila, Chlamydia

pneumoniae (also called the TWAR agent), and other rare agents.

1154A strong index of suspicion is required for diagnosis, especially in the

elderly and immunocompromised individuals, who have altered response

mechanisms. Subtle clues in the elderly include changes in mentation, confusion,

and exacerbation of other illnesses. The febrile response may be entirely absent,

and the results of the physical examination are not predictive of pneumonia. In

high-risk groups, an increased respiratory rate of greater than 25 breaths per

minute remains the most reliable sign of infection. Mortality in these high-risk

groups of patients is strongly correlated with the ability of the host to mount

normal defenses to the symptoms of fever, chills, and tachycardia.

All women suspected of having pneumonia should undergo chest

radiography to establish the diagnosis and to detect alternate diagnoses such

as congestive heart failure and tumors. [1] The chest radiograph can detect

complications like pleural effusions and multilobar disease. In the setting of CAP

in a markedly ill patient, a referral to a pulmonary specialist or to the local

emergency room may be indicated because of the high rate of severe

complications. The appropriate laboratory studies, including sputum cultures,

Gram stains, etc., can be obtained.

The American Thoracic Society updated their original guidelines in 2007 and

these are currently in the process of being revised again (12). These clinical

recommendations use an evidence-based approach for the diagnosis and

management of community-acquired pneumonia. Therapy should be directed at

the responsible or most likely pathogen (13), but in many cases of pneumonia, the

exact cause cannot be determined, and empiric therapy should be initiated. [1]

The American Thoracic Society recommends empiric therapy based on four

groups of specific patient profiles, the presence of modifying factors, and

pneumonia severity (Table 22-1):

Group I: Outpatients with no cardiopulmonary disease (congestive

heart failure or COPD) and no modifying factors. These patients are in

the lowest-risk group and are usually infected by pathogens such as C.

pneumoniae, M. pneumoniae, or S. pneumoniae. Patients should be treated

with an advanced-generation macrolide such as azithromycin,

clarithromycin, or doxycycline.

Group II: Outpatients with cardiopulmonary disease or modifying

factors. Patients in this group usually have some comorbidities and are

older than 50 years of age. Aerobic gram-negative bacilli, mixed infections

with atypical pathogens, and drug-resistant S. pneumoniae (DRSP) should

be considered in this patient population. Drug recommendations include a

respiratory fluoroquinolone (moxifloxacin, gemifloxacin, or levofloxacin)

or beta-lactam PLUS macrolide.

1155Group III: Inpatients who are not in the intensive care unit and have

cardiopulmonary or modifying factors. Drugs for these patients include

intravenous fluoroquinolone monotherapy or a combination of an

intravenous beta-lactam agent plus either intravenous or oral administration

of an advanced macrolide or doxycycline.

Group IV: Inpatients in the intensive care unit. These patients usually

have the most severe pneumonia, and all antibiotics are given

intravenously. Immediate consultation with an internist, hospitalist, or

infectious disease specialist is recommended.

Table 22-1 Modifying Factors that Increase the Risk of Infection with Specific

Pathogens

Penicillin-resistant and Drug-resistant Pneumococci

Age >65 yrs

Beta-lactam therapy within the past 3 mo

Alcoholism

Immune-suppressive illness (including therapy with corticosteroids)

Multiple medical comorbidities

Exposure to a child in a day-care center

Enteric gram-negatives

Residence in a nursing home

Underlying cardiopulmonary disease

Multiple medical comorbidities

Recent antibiotic therapy

Pseudomonas aeruginosa

Structural lung disease (bronchiectasis)

Corticosteroid therapy (>10 mg of prednisone per day)

Broad-spectrum antibiotic therapy for >7 days in the past month

Malnutrition

1156Adapted from American Thoracic Society. Guidelines for the management of adults with

community-acquired pneumonia. Am J Respir Crit Care Med 2001;163:1730–1754.

Oxygen therapy and hydration should be initiated in addition to antibiotic

therapy. Given issues of bacterial resistance and development of severe lifethreatening compromise, patients in groups III, IV, and the sicker patients in

group II may benefit from consultation with a pulmonary specialist or an internist.

Most patients will have an adequate clinical response within 3 days of treatment.

Oral antibiotics may be given when patients meet the following criteria: ability to

eat and drink, improvement in cough and dyspnea, afebrile (<100°F) on two

occasions 8 hours apart, and a decreasing white blood cell count. If other clinical

features are favorable, patients may be switched to oral antibiotics even if febrile.

They may be discharged on the same day that oral antibiotics are started if other

medical and social factors are favorable.

Vaccination

There are numerous vaccines that need to be administered to adults

depending on age, comorbidities, and presence of young children. All primary

care providers should be familiar with the recommended immunizations and urge

their patients to have them. Many are available at pharmacies by prescription if a

practice has not undertaken the cost of providing vaccines at the office. The

Centers for Disease Control and Prevention (CDC) has a comprehensive chart

outlining the vaccines for adults (14). See Figure 22-1. The influenza vaccine

should be given every fall to high-risk groups: individuals 50 years of age or

older; anyone with serious long-term health problems such as heart disease,

lung disease, kidney disease, diabetes, and weak immune systems as with

HIV and AIDS; individuals on long-term steroids or receiving cancer

treatment; women who are pregnant during the flu season (November

through April); and anyone coming in close contact with people at risk of

serious influenza like physicians, nurses, and family members. Vaccination is

best given from October to mid-November. Antiviral agents should not be used as

a substitute for vaccination but may be a useful adjunct. The four agents approved

for use in the United States are amantadine, rimantadine, zanamivir, and

oseltamivir. These drugs should be given within 2 days of the onset of symptoms

to shorten the duration of uncomplicated illness caused by influenza (15).

CARDIOVASCULAR DISEASE

The risk factors for coronary artery disease are presented in Table 22-2.

Central to treating cardiovascular disease is the control of contributing

1157diseases and risk factors through lifestyle modifications (Table 22-3). Aerobic

exercise protects against cardiovascular disease (16). Additional aspects of

prevention of myocardial disease, renal disease, and stroke include control of

hypertension, identification and control of diabetes and obesity, and control of

dietary fats, especially cholesterol, in susceptible individuals (Fig. 22-2).

Table 22-2 Major Risk Factors for Coronary Artery Disease

Age >55 for men and >65 for women

Family history of cardiovascular disease (men <55 yrs; women <65 yrs)

Physical inactivity

Diabetes mellitus

Cigarette smoking

Dyslipidemia

Obesity (body mass index ≥30)

Hypertension

Microalbuminuria or estimated glomerular filtration rate <60 mL/min

Adapted from Chobanian AV, Bakris GL, Black HR, et al. The seventh report of the

Joint National Committee on Prevention, Detection, Evaluation, and Treatment of High

Blood Pressure (JNC VII). JAMA 2003;289:2560–2572.

1158FIGURE 22-1 Recommended immunizations for adults by health condition 2017.

(Adapted from U.S. Department of Health and Human Services, Center for Disease

Control and Prevention. Recommended immunizations for adults by age. Available online

at https://www.cdc.gov/vaccines/schedules/downloads/adult/adult-schedule-easy-read.pdf.

Accessed September 28, 2017.)

1159FIGURE 22-2 Disease and risk factors contributing to cardiovascular disease.

Table 22-3 Lifestyle Adjustments to Manage Hypertension

Weight reduction to maintain a body mass index of 18.5–24.9

Limit alcohol use to two drinks per day for men (24 oz beer, 10 oz of wine, 3 oz of

80-proof whiskey) and no more than one drink per day for women and lighter-weight

persons

Regular aerobic exercise (at least 30 min per day of brisk walking most days of the

week)

Decrease salt intake to less than 2.4 g of sodium or 6 g of sodium chloride per day

Consume a diet rich in fruits, vegetables, and low-fat dairy products with a reduced

content of saturated and total fat

Adapted from Chobanian AV, Bakris GL, Black HR, et al. The seventh report of the

Joint National Committee on Prevention, Detection, Evaluation, and Treatment of High

Blood Pressure (JNC VII). JAMA 2003;289:2560–2572.

Hypertension

The relationship between hypertension and cardiovascular events such as

stroke, coronary artery disease, congestive heart disease, and renal disease is

well known. More than 50 million people in the United States have

1160hypertension. It is found in 15% of the population between the ages of 18 and 74

years; the incidence increases with age and varies with race. Recognition and

treatment of hypertension may decrease the development of renal and cardiac

disease.

Epidemiology

The incidence of hypertension is twice as high in African Americans than in

whites. Geographic variations exist: the southeastern United States has a higher

prevalence of hypertension and stroke, regardless of race (17). Preventive

measures can be most effective in those at highest risk, such as in African

American women and individuals from the lowest socioeconomic level (18). The

influence of genetic predisposition is poorly understood. Classically,

hypertension is defined as blood pressure levels higher than 140/90 when

measured on two separate occasions. Life insurance risk tables indicate that

when blood pressure is controlled to lower than 140/90, normal survival occurs

over a 10- to 20-year follow-up, regardless of gender. Recommendations are

based on sustained blood pressures higher than 140/90 (see Fig. 22-3) (19).

Table 22-4 Laboratory Tests and Procedures Recommended in the Evaluation of

Uncomplicated Hypertensiona

Urinalysis

Complete blood count

Potassium

Creatinine or estimated glomerular filtration rate

Calcium

Fasting glucose

Lipid profile that includes HDL, LDL, and triglycerides after a 9- to 12-hr fast

12-lead electrocardiogram

aIf any of the above are abnormal, consultation or referral to an internist is indicated.

HDL, high-density lipoprotein; LDL, low-density lipoprotein.

Adapted from Chobanian AV, Bakris GL, Black HR, et al. The seventh report of the

Joint National Committee on Prevention, Detection, Evaluation, and Treatment of High

Blood Pressure (JNC VII). JAMA 2003;289:2560–2572.

1161Table 22-5 Blood Pressure (BP) Classification (Adults 18 Yrs and Older)

Category Systolic BP (mm Hg) Diastolic BP (mm Hg)

Normal <120 and <80

Prehypertension 120–139 or 80–89

Stage 1 hypertension 140–159 or 90–99

Stage 2 hypertension >160 or >100

Modified from Chobanian AV, Bakris GL, Black HR, et al. The seventh report of the

Joint National Committee on Prevention, Detection, Evaluation, and Treatment of High

Blood Pressure (JNC VII). JAMA 2003;289:2560–2572.

More than 95% of individuals with hypertension have primary or essential

hypertension (cause unknown), whereas fewer than 5% have secondary

hypertension resulting from another disorder. [2] Key factors to be determined

in the history and physical examination include presence of prior elevated

readings including a history of pre-eclampsia, previous use of antihypertensive

agents, a family history of cardiovascular death before age 55, use of weight-loss

supplements and excessive intake of alcohol or sodium (Tables 22-2 and 22-3).

Lifestyle modification is considered important in the therapy of hypertension;

thus, a detailed history of diet and physical activity should be obtained (16).

Baseline laboratory evaluations to rule out reversible causes of hypertension

(secondary hypertension) are listed in Table 22-4. Diagnosis and management are

based on the classification of blood pressure readings, as presented in Table 22-5.

The Joint National Committee on Prevention, Detection, Evaluation, and

Treatment of High Blood Pressure (JNC7) released their seventh report in 2003.

The purpose was to provide an evidence-based approach to the prevention and

management of hypertension. [2] Following are some of the key points of this

report:

Systolic blood pressure in those older than 50 years is a more

important cardiovascular risk factor than diastolic blood pressure.

Beginning at 115/75 mm Hg, the risk of cardiovascular disease doubles

for each increment of 20/10 mm Hg.

Individuals who are normotensive at 55 years of age will have a 90%

lifetime risk of developing hypertension.

Patients with prehypertension (systolic blood pressure 120 to 139 mm

Hg or diastolic blood pressure 80 to 89 mm Hg) require health-

1162promoting lifestyle modifications to prevent the progressive rise in

blood pressure and cardiovascular disease.

For uncomplicated hypertension, thiazide diuretic should be used in

most cases for medical treatment, either alone or combined with drugs

from other classes.

Other antihypertensive drug classes (ACE inhibitors, angiotensinreceptor blockers, beta blockers, calcium channel blockers) should be

used in the presence of specific high-risk conditions (Fig. 22-3).

These recommendations were supplemented in the 2014 JNC8 meeting

with the following (19):

In the general population aged 60+, initiate pharmacologic treatment at

systolic pressures ≥150 mm Hg or diastolic blood pressure ≥90 mm Hg to

reach treatment goal of less than 150/90 mm Hg.

In the general population aged less than 60, initiate pharmacologic

treatment to lower blood pressure at a diastolic of 90 mm Hg or greater.

In the general population aged less than 60, initiate pharmacologic

treatment to lower blood pressures at a systolic of 140 mm Hg or greater.

In population aged 18 or more with chronic kidney disease or diabetes,

initiate pharmacologic treatment to lower blood pressure at systolic blood

pressure of 140 mm Hg or greater or diastolic blood pressure of 90 mm Hg

or greater.

In the general black population including those with diabetes, initial

antihypertensive treatment should include a thiazide-type diuretic or

calcium channel blocker.

The main objective of hypertensive treatment is to attain and maintain a

goal BP. If the goal BP is not reached within a month of treatment, increase

the dose of the first drug or add a second agent. Referral to a hypertension

specialist may be indicated for patients in whom goal BP cannot be attained

using the above strategies or for the management of complicated patients.

[2] Regardless of therapy or care, hypertension will be controlled only if patients

are motivated to maintain their treatment plan. If blood pressure control is not

easily achieved, if the systolic blood pressure is higher than 180 mm Hg, or if the

diastolic reading is higher than 110 mm Hg, referral to an internist is

recommended. Referral is indicated if secondary hypertension is suspected or

evidence of end-organ damage (renal insufficiency or congestive heart failure) is

present.

Measurement of Blood Pressure

1163Essential variables in the evaluation of hypertension are the acquisition of

measurements and the need to standardize measurements (20). “White coat”

or office hypertension (i.e., elevated just by seeing a physician) may occur in

up to 30% of patients. For patients who have repeated normal measures outside

of the office, it is reasonable to use ambulatory or home monitoring devices.

Given the variation of accuracy and patient interpretation, it is advisable for the

patient to bring their blood pressure unit into the office to calibrate it against the

office-based measurements.

Blood pressure protocols for measurement should be standardized. The

following steps will optimize the accuracy of the reading:

The patient should rest for 5 minutes in a seated position with legs

uncrossed.

Use the right arm for measurements (for unknown reasons, the right arm

has higher readings).

The cuff should be applied 2 cm above the bend of the elbow.

The cuff should be inflated to 30 mm Hg above the disappearance of the

brachial pulse, or 220 mm Hg.

The cuff should be deflated slowly. The cuff size is important, and most

cuffs are marked with “normal limits” for the relative size they can

accommodate. The most common clinical problem encountered is small

cuffs used with obese patients, resulting in “cuff hypertension.”

Phase-V Korotkoff is when sounds completely disappear. Most experts in

hypertension advocate the use of phase-V Korotkoff sounds.

The use of automated devices may help eliminate discrepancies in

measurements. Regardless of the method or device used, two measurements

should be obtained with less than a 10 mm Hg disparity to be judged adequate.

When repeated measures are performed, there should be a 2-minute rest period

between readings. Blood pressure has a diurnal pattern, so determinations

preferably should be done at the same time.

Therapy

[2] Nonpharmacologic interventions or lifestyle modifications should be

attempted before initiation of medication. Drug therapy should be initiated

for systolic blood pressure greater than 140 mm Hg or diastolic blood

pressure greater than 90 mm Hg. An important element in lifestyle

modifications is to modify all contributors to cardiovascular disease. In obese

patients, weight loss, especially in individuals with truncal and abdominal

obesity, can play a significant role in the prevention of atherosclerosis (16). A

1164loss of just 10 lb was reported to lower blood pressure. Enquiries into dietary

practices should be made to eliminate excess salt, cholesterol, and fats in the diet.

Dietary interventions that use calcium, magnesium, and potassium

supplementation did not make a clinically significant reduction in pressure (21).

[2] An exercise program, weight loss, and moderating alcohol intake (to no

more than two alcoholic beverages per day) contribute to overall

cardiovascular health. Aerobic exercise alone may prevent hypertension in

20% to 50% of normotensive individuals (16).

[2] The goal of therapy is for the patient to lower blood pressure into the

“normal range”: a systolic reading less than or equal to 120 mm Hg and a

diastolic reading less than or equal to 80 mm Hg. If lifestyle modifications

are not sufficient to control blood pressure, then pharmacologic intervention

is indicated (Fig. 22-3).

Diuretics

The most commonly used medication for initial blood pressure reduction is a

thiazide diuretic. The mechanism of action is to reduce plasma and extracellular

fluid volume. This lowering of volume is thought to decrease peripheral

resistance. Cardiac output initially decreases and then normalizes (19). The

important long-term effect is a slight decrease in extracellular fluid volume.

Potassium-sparing diuretics (spironolactone, triamterene, or amiloride) are

available in fixed doses and should be prescribed to prevent the development of

hypokalemia. Potassium supplementation is less effective than the use of

potassium-sparing agents. Thiazide diuretics are best used in patients with

creatinine levels less than 2.5 g/L. Control of hypertension with concurrent renal

insufficiency is difficult and is probably best handled by an internist or

nephrologist. Concurrent use of nonsteroidal anti-inflammatory drugs (NSAIDs)

limits the effectiveness of this class of drugs. Other side effects of thiazide

diuretics include hyperuricemia, which may contribute to acute gout attacks,

glucose intolerance, and hyperlipidemias (19).

Angiotensin-Converting Enzyme Inhibitors

The ACE inhibitors are first-line drugs in the treatment of hypertension.

There are relatively few side effects; chronic cough is the most worrisome and is

a common reason of discontinuing the use of this group of drugs. Other agents

should be considered for patients at risk for pregnancy (a strict contraindication).

ACE inhibitors can be used in combination with other agents, including diuretics

and calcium channel antagonists. In contrast to beta-blocking agents, these

medications can be used in patients with asthma, depression, and peripheral

vascular disease. For unknown reasons, they are less effective in African

1165Americans unless a diuretic is used concomitantly. Use with diuretics increases

the effectiveness of both drugs, but hypovolemia may result and must be

monitored. Any NSAID, including aspirin, may decrease the antihypertensive

effectiveness. Creatinine levels should be measured at the start of therapy

and 1 week after initiation of any ACE inhibitor. An increase of up to 35% of

the baseline creatinine value is acceptable, and treatment should be continued

unless hyperkalemia develops.

Angiotensin-Receptor Blockers

The angiotensin-receptor blockers such as losartan and valsartan interfere

with the binding of angiotensin II to AT1 receptors. As with ACE inhibitors,

they are effective in lowering blood pressure, without causing the side effect

of coughing. Angiotensin-receptor blockers have favorable effects on the

progression of kidney disease in individuals who have diabetes, and on those

without diabetes and congestive heart failure.

Calcium-Channel Blockers

Calcium-channel blockers represent a major therapeutic breakthrough for

patients with coronary artery disease. They are effective in patients with

hypertension and peripheral vascular disease. The mechanism of action is to

block calcium movement across smooth muscle, therefore promoting vessel wall

relaxation. Calcium channel blockers are useful in treating concurrent

hypertension and ischemic heart disease. In addition, these drugs are particularly

effective in the elderly and African Americans. Side effects noted include

headache, dizziness, constipation, gastroesophageal reflux, and peripheral edema.

The addition of long-acting calcium-channel blockers made these preparations

more amenable for use in hypertension. A relative contraindication for use of

these drugs is the presence of congestive heart failure or conduction disturbances.

Adrenergic Inhibitors

Beta blockers were used extensively for years as antihypertensive agents. The

mechanism of action is decreasing cardiac output and plasma renin activity, with

some increase in total peripheral resistance. As a class, they are an excellent

source of first-line therapy, especially for migraine sufferers. Formulations such

as atenolol are water soluble, beta1 selective, and have fewer side effects than

propranolol. At higher doses, beta2 effects emerge. An advantage of watersoluble agents is a longer half-life. Reduced dosing schedules improve

compliance. Side effects of beta blockers include an increase in triglyceride levels

and a decrease in high-density lipoprotein (HDL) cholesterol and blunting of

1166adrenergic release in response to hypoglycemia. NSAIDs may decrease the

effectiveness of beta blockers. Contraindications to beta blockers are asthma, sick

sinus syndrome, or bradyarrhythmia.

The use of alpha1-adrenergic drugs as single agents decreases total

cholesterol and low-density lipoprotein (LDL) cholesterol while increasing HDL

cholesterol, in contrast to the metabolic effects of beta-blocking agents. They may

contribute to stress urinary incontinence in women because of altered urethral

tone. Their mode of action is to promote vascular relaxation by blocking

postganglionic norepinephrine vasoconstriction in the peripheral vascular smooth

muscle. When alpha1-adrenergic drugs are used in combination with diuretics,

hypotension may be further exacerbated. Therapy should begin with small doses

taken at bedtime followed by incremental increases. Other side effects that may

limit the usefulness of these agents in some patients include tachycardia,

weakness, dizziness, and mild fluid retention.

Direct Vasodilators

Hydralazine is a potent vasodilator used for years in obstetrics for severe

hypertension associated with preeclampsia and eclampsia. The mechanism of

action is direct relaxation of vascular smooth muscle, primarily arterial. Major

side effects include headaches, tachycardia, and fluid (sodium) retention that may

result in paradoxical hypertension. Several drug combinations are used to counter

the side effects and enhance antihypertensive effects of hydralazine. This is not a

typical first line medication.

Central-Acting Agents

Central-acting agents (methyldopa and clonidine) have long been used in

obstetrics. The mechanism of action is to inhibit the sympathetics in the central

nervous system, resulting in peripheral vascular relaxation. Side effects, including

taste disorders, dry mouth, drowsiness, and the need for frequent dosing (except

for the transdermal form of clonidine), limited the popularity of this group of

drugs. Sudden withdrawal of clonidine may precipitate a hypertensive crisis

and induce angina. Compliance is always a major issue, and side-effect profiles

contribute significantly to patient nonadherence. With the introduction of new

classes of drugs with improved efficacy and reduced side effects, the use of

medications in this class is expected to decline.

Monitoring Therapy

Blood pressure readings should be monitored frequently by the patient, or in

the office at 1- to 2-week intervals, when initiating intervention. If the patient

has other diseases (i.e., cardiovascular, renal), therapy should be initiated earlier

1167and directed to the target organ. If lifestyle modification alone is successful, close

monitoring is necessary at 3- to 6-month intervals. When lifestyle modification is

unsuccessful, a blood pressure medication should be started to decrease target

organ disease. When beginning therapy, concurrent medical conditions treatable

with a common agent should be sought. Gender is not an important consideration

in choosing an antihypertensive agent. However, presence of diabetes, renal

disease, or race can impact preferred initial medication. Figure 22-3 shows a

schematic of how to approach initiating pharmacologic interventions.

After antihypertensive medications are initiated, monitoring should be

instituted at approximately monthly intervals to determine blood pressures

and to assess side effects. The serum creatinine and potassium levels should be

monitored one to two times per year. When blood pressure goals are reached,

patients may be seen in the office at 3- to 6-month intervals. Patients capable of

home blood-pressure monitoring should be encouraged to measure the blood

pressure at the same time twice weekly. If intolerable side effects develop, a

different class of medications should be used and the patient’s progress

monitored. Patients whose blood pressure is difficult to control, especially if

requiring two agents, should be considered for referral. Patients with evidence of

target organ disease should be considered for referral to the appropriate specialist

for more intensive diagnostic workup and therapy.

Cholesterol

[3] The dietary influence of cholesterol on atherosclerosis and its relationship

to hypertension and cardiovascular events (myocardial infarction and

stroke) is widely debated in the scientific and lay communities. The

controversy centers on the effect of dietary cholesterol in assessing the risk

and prevention of cardiovascular disease (22). Many assume that all

cholesterol and fat in the diet have negative health consequences. Cholesterol

metabolism is complex, and some of our knowledge is extrapolated from animal

models. The role of cholesterol testing (who, when, and at what age) is hotly

debated among health care professionals, and the test itself is fraught with

multiple variables that affect results.

1168FIGURE 22-4 Metabolic pathways of lipid metabolism. Apo, apoprotein; LP, lipoprotein;

FFA, free fatty acid; IDL, intermediate-density lipoprotein; LDL, low-density lipoprotein;

VLDL, very–low-density lipoprotein; HDL, high-density lipoprotein; LCAT, lecithin

cholesterol acyltransferase.

Terms and Definitions

Cholesterol is usually found in an esterized form with various proteins and

glycerides that characterize the stage of metabolism. The important lipid particles

in cholesterol metabolism are noted in the schematic on Figure 22-4.

Metabolism

Cholesterol metabolism is divided into two pathways: (i) the exogenous

pathway derived from dietary sources, and (ii) the endogenous pathway or

the lipid transport pathway. Individuals vary in their ability to metabolize

1169cholesterol. Hyporesponders may be given cholesterol-loaded diets with no effect

on serum cholesterol measurements. Hyperresponders, in contrast, have high

serum cholesterol levels, regardless of dietary intake. Explanations for these

differences are well described in animal models, but not in humans.

Despite the negative connotation of LDL in cardiovascular disease, it is a very

important cellular metabolite and precursor for adrenocortical cells, lymphocytes,

and renal cells. The liver uses LDL for synthesis of bile acids and free cholesterol,

which is secreted into the bile. In the normal human, 70% to 80% of LDL is

removed from the plasma each day and secreted in the bile by utilization of the

LDL receptor pathway.

The final metabolic pathway is the transformation of HDL cholesterol in the

extrahepatic tissue. HDL cholesterol carries the plasma enzyme lecithin

cholesterol acyltransferase (LCAT). LCAT allows HDL cholesterol to

resynthesize lipids to very–low-density lipoprotein (VLDL) cholesterol and

recycle the lipid cascade. HDL cholesterol acts as a “scavenger” and therefore

reverses the deposit of cholesterol into tissues. There is good evidence that HDL

cholesterol is responsible for the reversal of atherosclerotic changes in vessels,

hence the term “good cholesterol” (22).

Hyperlipoproteinemia

When cholesterol is measured, various fractions are reported. Plasma cholesterol

or total cholesterol consists of cholesterol and unesterified cholesterol fractions. If

triglycerides are analyzed in conjunction with cholesterol, then assumptions can

be made concerning which metabolic pathway may be abnormal.

Hyperlipoproteinemias are defined by establishing a “normal population”

and then setting various limits at the 10th and 90th percentiles. Standards

for women set the 80th percentile for cholesterol at 240 mg/dL and the 50th

percentile at 200 mg/dL (Table 22-6). A diet low in animal fat and high in

vegetable and fiber consumption helps control the level of cholesterol. Plasma

elevations of chylomicrons, LDL, VLDL, various remnants of intermediatedensity lipoprotein (IDL), and VLDL are classified by the elevated fraction.

Evaluation

There are multiple causes of variation in cholesterol measurements (23). [3]

Major sources of variation within individuals include diet, obesity, smoking,

ethanol intake, and the effects of exercise. Other clinical conditions that affect

cholesterol measurements include hypothyroidism, diabetes, acute or recent

myocardial infarction, and recent weight changes. Measurements can be altered

by fasting, position of the patient while the sample is drawn, the use and duration

of venous occlusion, various anticoagulants, and the storage and shipping

1170conditions.

Table 22-6 Initial Classification Based on the Total Cholesterol, LDL, HDL, and

Triglyceride Levels

Initial Classification

Total cholesterol

<200 mg/dL Desirable blood cholesterol

200–239 mg/dL Borderline high blood cholesterol

≥240 mg/dL High blood cholesterol

LDL cholesterol

<100 mg/dL Optimal cholesterol

100–129 mg/dL Near or above optimal

130–159 mg/dL Borderline high

160–189 mg/dL High

≥190 mg/dL Very high

HDL cholesterol

<40 mg/dL Low HDL cholesterol

≥60 mg/dL High HDL cholesterol

Triglycerides

<150 mg/dL Normal

150–199 mg/dL Borderline high

200–499 mg/dL High

>500 mg/dL Very high

HDL, high-density lipoprotein; LDL, low-density lipoprotein.

Adapted from Expert Panel on Detection, Evaluation, and Treatment of High Blood

Cholesterol in Adults. Executive summary of the third report of the National Cholesterol

Education Program (NCEP) Expert Panel on the Detection, Evaluation, and Treatment of

1171High Blood Cholesterol in Adults. JAMA 2001;285:2486–2497.

Age and gender contribute to variations in total cholesterol

measurements. [3] Before age 50, women have lower lipid values than

men, after which age the level in women is higher than in men. This

finding may be modified by exogenous oral conjugated estrogens.

Seasonal variation also occurs, with lipid samples in December or

January being found to be approximately 2.5% higher than those measured

in June or July.

The effect of diet and obesity is well established. [3] Weight reduction in

an obese individual affects the triglyceride level, which may decrease as

much as 40%. Total cholesterol and LDL decrease less than 10% with diet;

however, HDL increases approximately 10%. Weight gain negates any

benefit from prior weight loss. Accuracy of lipid measurements depends on

the stability of the patient’s weight.

Alcohol and cigarette smoking are well-known modifiers of cholesterol.

Moderate sustained alcohol intake increases HDL and decreases LDL;

there is a complementary increase in triglycerides. [3] Alcohol has a

protective effect when taken in moderation (defined as approximately

two alcoholic drinks [2 oz of absolute alcohol] per day), but this effect

is negated in higher quantities. Smoking has the opposite effect,

increasing LDL and triglyceride levels and decreasing HDL. HDL3

decreases with cigarette smoking. The critical number of cigarettes smoked

is 15 to 20 per day, regardless of gender, and a variation in the number

smoked will affect results. Caffeine has a mixed effect on lipoprotein

measurements and should be avoided for 12 hours before blood collection.

Exercise is an important variable in the overall risk management of

heart disease. [3] Moderate levels of exercise are as important in the

overall cardiovascular health as control of hypertension and cessation of

cigarette smoking. Strenuous exercise lowers the concentrations of

triglycerides and LDL and increases HDL in the serum. Because of these

acute blood changes, vigorous exercise should be avoided within 12 hours

of drawing the blood for testing.

Patients with hypothyroidism have increased levels of total cholesterol

and LDL.

Testing

Because of the diurnal variation of blood triglycerides, blood samples should

be collected in the morning after a 12-hour fast. One of the most important

aspects of overall standardization of lipoprotein measurements is the laboratory

1172used. It may be worthwhile to consult a clinical pathologist to determine if the

laboratory complies with CDC standards for cholesterol and lipoprotein

measurements.

Management

When hyperlipidemia is confirmed on at least two separate occasions, secondary

causes should be diagnosed or excluded by taking a detailed medical and drug

history, comprehensive physical examination, and appropriate laboratory tests.

Causes of secondary dyslipidemia include diabetes, hypothyroidism, obesity,

obstructive liver disease, chronic renal failure, pregnancy, and use of medications

such as progestins, anabolic steroids, and corticosteroids. Therapeutic lifestyle

changes should be initiated in all patients to reduce their risk of coronary

heart disease:

1. [3] Reduced intakes of saturated fats (<7% of total calories) and

cholesterol (<200 mg per day)

2. Therapeutic options for enhancing LDL lowering, such as plant

stanols/sterols 2 g per day and increased viscous (soluble) fiber 10 to 25 g

per day

3. Weight reduction

4. Increased physical activity

5. Smoking cessation and alcohol only in moderation

The 2013 ACC/AHA Cholesterol Management guidelines changed the

management of cholesterol to prevent the occurrence of cardiovascular disease

including stroke (24). The recommendations primarily involved patient age,

family history of hypercholesterolism, gender, and presence of comorbidities,

along with lipid levels. To assist in judging individual risks, an atherosclerotic

cardiovascular disease (ASCVD) risk calculator has been developed by the AHA

(25). Although many groups challenge the accuracy of the calculations stating

they consistently overestimate risks, it is still a useful tool.

[3] The level I recommendations from the 2013 guidelines regarding initiation of

medication included:

High-intensity statin therapy should be initiated (or continued) in patients

≤75 with clinical ASCVD. If not tolerated, moderate-intensity therapy is

second line.

Individuals with LDL ≥190 mg/dL or triglycerides ≥500 need to be

evaluated for secondary causes of hyperlipidemia.

Adults >21 with LDL >190 mg/dL should be treated with statins (high

1173intensity if tolerated).

Moderate-intensity statin therapy should be initiated (continued) for adults

aged 40 to 75 years with diabetes.

ASCVD calculator should be used to estimate 10-year ASCVD risk for

individuals with LDL 70 to 189 mg/dL without clinical ASCVD to guide

when statins should be initiated.

Adults 40 to 75 years of age with LDL 70 to 189 mg/dL without clinical

ASCVD or diabetes and an estimated 10-year risk of ASCVD ≥7.5%

should be treated with moderate-intensity statins.

[3] Patients with a family history of cardiovascular disease (history of

premature coronary artery problems and strokes) should be tested and

started on conservative programs in their 20s. As noted above, if their LDL

is greater than 190 mg/dL, they should be started on statins. Otherwise an

ASCVD calculation should be done and pharmaceutical therapy started if the 10-

year risk is 7.5% or more. Any woman with coronary heart disease or equivalents

such as diabetes or other forms of atherosclerotic disease (peripheral arterial

disease, abdominal aortic aneurysm, and symptomatic carotid artery disease)

should initiate lifestyle changes if her LDL is 100 mg/dL or more and drug

therapy if her LDL is 190 mg/dL or her 10-year risk calculation is 7.5% or more.

Periodic assessment of cardiovascular risk factors should be done starting at

age 40 in patients without prior identified risks. An annual assessment of weight,

blood pressure, exercise routine, and smoking status is supported by expert

opinion. A true screen requires lipid profile. Recommendations are to do this

every 5 years unless there is a significant change in the patient’s risk profile,

which may merit more frequent screens. The data for routine screening in patients

less than age 40 is unclear with no study clearly demonstrating a benefit. For

these reasons, USPSTF states it can make no recommendation for or against such

screening (26).

Prior to the 2013 ACC/AHA guidelines and confirmed by the U.S. Preventive

Service Task Force recommendation, bile acid–binding resins cholestyramine and

colestipol were the mainstay of therapy (26). The significant side effects of

nicotinic acid and fibric acid derivatives and poor patient compliance caused by

those side effects relegated them to second or third line treatment.

[3] Statins (HMG-CoA [3]-hydroxy-3methyl-glutaryl-coenzyme A reductase

inhibitors) have become the mainstay of treatment and prevention. These include

atorvastatin, fluvastatin, lovastatin, pravastatin, and simvastatin. These

medicines inhibit HMG-CoA reductase, the enzyme that catalyzes the ratelimiting step in cholesterol synthesis. Multiple clinical trials showed that

pravastatin, simvastatin, and lovastatin have a beneficial effect in

1174cardiovascular disease. Statins are better tolerated than other lipid-lowering

drugs, but reported side effects have concerned patients. These include severe

myalgias, muscle weakness with increases in creatine phosphokinase, and, rarely,

rhabdomyolysis, leading to renal failure. Detailed studies have shown that most of

these are mild and resolve with cessation of the medication (24,26,27). The severe

side effects of rhabdomyolysis and renal failure are extremely rare. This results in

a very favorable benefit to risk ratio for the statins when used in a moderate-risk

population (27). As the 10-year risk decreases, the benefit to risk ratio also

decreases. For this reason, the USPSTF recommends that patients with less than a

10% risk of an ASCVD event in the next 10 years not start statins without a

physician/patient discussion of risks and benefits of statins.

DIABETES MELLITUS

DM is a chronic disorder of altered carbohydrate, protein, and fat metabolism

resulting from a deficiency in the secretion or function of insulin. The disease is

defined by the presence of either fasting hyperglycemia or elevated plasma

glucose levels based on an oral glucose tolerance testing (OGTT). The major

complications of DM are primarily vascular, renal, and metabolic. [4] The

prevalence of DM is higher in women (especially with a history of gestational

diabetes) and certain ethnic groups, although a background rate in the general

population is 6.29%, which has increased threefold in 15 years (28).

[4] Risk factors for DM are:

1. Age greater than 45 years

2. Adiposity or obesity

3. A family history of diabetes

4. Race/ethnicity

5. Hypertension (blood pressure 140/90 mm Hg or greater)

6. HDL cholesterol less than or equal to 35 mg/dL and/or a triglyceride level

greater than or equal to 250 mg/dL

7. History of gestational diabetes or delivery of a baby weighing more than 9

lb

Major complications of DM include blindness, renal disease, gangrene of an

extremity, heart disease, and stroke. Diabetes is one of the four major risk factors

for cardiovascular disease.

Classification

In 2016, an expert committee was convened by the American Diabetes

1175Association to review the proposed standards for medical care in diabetes. Their

findings were reported in 2017 in Diabetes Care. The goal of the revision was to

clarify guidelines for nomenclature and testing that might reduce diagnostic

confusion and improve patient well-being (Table 22-7). The terms insulindependent diabetes mellitus (IDDM) and noninsulin-dependent diabetes mellitus

(NIDDM) were replaced by the terms type 1 and type 2 DM based on insulin

levels and function but not on the patient’s age.

Type 1 Diabetes Mellitus

With type 1 diabetes, the major metabolic disturbance is the absence of

insulin from the destruction of beta cells in the pancreas. Insulin is necessary

for glucose metabolism and cellular respiration. When insulin is absent, ketosis

results. The cause of type 1 diabetes is unknown; data suggest an autoimmune

association from either a viral infection or toxic components in the environment.

Studies in the past decade showed a correlation between many autoimmune

diseases and the human leukocyte antigens (HLA).

Table 22-7 Classification of Diabetes Mellitus

1. Type 1 diabetes

Characterized by pancreatic destruction leading to insulin deficiency typically due to

autoimmune beta cell destruction

2. Type 2 diabetes

A combination of insulin resistance and some degree of inadequate insulin secretion

3. Gestational diabetes mellitus

Is diabetes diagnosed in the second or third trimester of pregnancy without preexisting diabetes

4. Specific types of diabetes due to other causes

A. Endocrinopathies (Cushing, acromegaly, pheochromocytoma,

hyperaldosteronism)

B. Drug- or chemical-induced (esp. organ transplant medications or glucocorticoids)

C. Diseases of the exocrine pancreas (pancreatitis, neoplasia, cystic fibrosis)

D. Infections

E. Genetic defects of beta-cell function and insulin action

Adapted from Cefalu W, ed. Standards of medical care in diabetes—2017. Diabetes Care

2017;40(supplement 1).

Insulin-sensitive tissues (muscle, liver, and fat) fail to metabolize glucose

efficiently in the absence of insulin. In uncontrolled type 1 diabetes, an excess

1176of counter-regulatory hormones (cortisol, catecholamines, and glucagon)

contributes to further metabolic dysfunction. In the absence of adequate amounts

of insulin, increasing breakdown products of muscle (amino acid proteolysis), fat

(fatty acid lipolysis), and glycogen (glucose glycogenolysis) are recognized.

There is an increase in glucose production from noncarbohydrate precursors as a

result of gluconeogenesis and ketogenesis in the liver. Without prompt treatment,

severe metabolic decompensation (i.e., diabetic ketoacidosis) will occur and may

lead to death.

Given the significant complexity and risks involved in the management of type

I DM, it is not advised that a generalist be primarily responsible for the

management of insulin and the associated comorbidities. These patients should be

followed by a provider who specializes in diabetes management.

Type 2 Diabetes Mellitus

[4] Type 2 DM is a heterogeneous form of diabetes that commonly occurs in

older age groups (>40 years) and more frequently has a familial tendency

than type 1 diabetes. This form of DM accounts for approximately 90% to 95%

of those with diabetes. The presence of risk factors strongly influences the

development of type 2 diabetes in susceptible populations.

[4] Risk factors for type 2 diabetes include ethnicity, obesity, family history

of DM, sedentary lifestyle, impaired glucose tolerance (IGT), upper-body

adiposity, and a history of gestational diabetes and hyperinsulinemia.

In contrast to the absence of insulin that occurs with type 1 diabetes, in

type 2 diabetes the altered metabolism of insulin results in insulin resistance.

[4] This condition is characterized by impaired glucose uptake in target tissues. A

compensatory increase in insulin secretion results, causing higher-than-normal

circulating insulin levels (29). Obesity is present in 85% of affected patients. The

cause of type 2 diabetes is unknown, but defects in the secretion and action of

insulin are suspected.

Diagnosis

Three methods are available to diagnose DM in nonpregnant women:

1. A single fasting blood glucose greater than or equal to 126 mg/dL on two

separate occasions

2. An A1c ≥6.5% or random blood glucose equal to or above 200 mg/dL in

an individual with classic signs and symptoms of diabetes (polydipsia,

polyuria, polyphagia, and weight loss)

A 2-hour OGTT greater than or equal to 200 mg/dL after a 75-g load of

1177glucose. [4] The term IGT has been replaced with the term prediabetic state

and is not considered diabetes diagnosis. However, it is important to identify

these individuals for more frequent screening and intervention. Diagnostic

criterion for prediabetes is fasting glucose greater than or equal to 100

mg/dL but less than 126 mg/dL, or A1c between 5.7% and 6.4%, or a 2-hour

value on a 75-g OGTT between 140 and 199 mg/dL (29).

It should be noted that fasting blood glucose, 2-hour OGTT, and A1c

screenings perform similarly but interestingly often pick up different patients with

positive screens. The 2-hour OGTT will result in the largest number of patients

receiving a diagnosis of diabetes. A1c is often the easiest initial screen but the

results can be impacted by race/ethnicity and anemia/hemoglobulinopathies.

[4] Patients who should be considered for diabetes testing can be

determined by the use of a diabetes risk calculator or using a listing of risk

factors. The calculators can be found at the American Diabetes Association

website and are available for downloads (30). Historical risk factors include:

All individuals 45 years of age or older (repeat at a minimum of 3-year

intervals)

Persons with classic signs and symptoms of diabetes (i.e., polyuria,

polydipsia, polyphagia, and weight loss)

Ethnic groups at high risk (Pacific Islanders, Native Americans,

African Americans, Hispanic Americans, and Asian Americans)

Obesity or overweight (body mass index >25 kg/m2) (or 23 kg/m2 if

Asian American)

History of a first-degree relative with diabetes

Women with gestational diabetes or who have delivered a baby

weighing more than 9 lb

Individuals with hypertension (blood pressure >140/90 mm Hg), or on

treatment for HBP or have a history of CVD

An HDL cholesterol level less than or equal to 35 mg/dL or triglyceride

level greater than or equal to 250 mg/dL

Presence of IGT/prediabetes on previous testing

Women with PCOS or other conditions associated with insulin

resistance.

Table 22-8 Generalist Physician Guidelines in the Therapy of Type II Diabetes

Mellitus

• Establish diagnosis and classify the type of diabetes mellitus (DM) (if type I, refer to

specialist in diabetes).

1178• Initiate diabetes education classes to learn blood glucose monitoring and diabetes

medications; to learn signs, symptoms, and complications; and to learn how to

manage sick days (may be available through local hospital or insurance plan).

• Place patient on ADA diet with appropriate caloric, sodium, and lipid restrictions

with aid of nutritionist or diabetologist to help with education and support.

• Establish baseline cardiac and renal risk factors, check feet and toenails at least once

a year, and refer to a foot specialist.

• Use finger-stick blood glucose for daily diabetic control.

• Follow chronic glycemic control by HgA1c every 2 to 3 mo in the office.

• Initial general health evaluation should consist of a complete history and physical

examination and the following laboratory tests: CBC with differential, chemistry

profile, lipid profile, urinalysis, thyroid function tests, urine for microalbuminuria,

and ECG (baseline at age 40 or older, repeat yearly).

• Development of vascular, ocular, neurologic, or renal compromise should prompt

immediate referral.

• Oral hypoglycemic agents may be considered if fasting blood glucose does not

decline or increases despite lifestyle changes. While on oral hypoglycemic agents,

check the HgA1C every 3 mo and at least two times a year if stable.

• If the fasting serum glucose is >200 mg/dL consistently or the HgA1C is more than

10%, consider starting insulin and referring the patient to an internist.

• Administer the flu vaccine every fall and the pneumococcal vaccine every 6 yrs.

ADA, American Diabetic Association; HgA1c, hemoglobin A1C; CBC, complete blood

count; ECG, electrocardiogram.

Adapted from Cefalu W, ed. Standards of medical care in diabetes—2017. Diabetes Care

2017;40(supplement 1).

Assessment of Glycemic Control

The only acceptable method for assessment of glycemic control is

determination of blood glucose by direct enzyme analysis. Glucometers with

memory storage made home glucose monitoring more reliable. Physician

treatment guidelines are in Table 22-8.

1179Treatment

Despite clear treatment recommendations, most diabetic patients have not reached

goals regarding A1c, LDL, and BP levels. Many continue to smoke and/or not

exercise. The reasons for the lack of success are complex, as is the care for most

patients with a chronic disease, especially those with a large behavioral

component. If a patient is not reaching goals through lifestyle adjustments and

oral medications, referral to a clinic system set up to deal with the multiple facets

of care should be made (29).

[4] Patients with prediabetes should be encouraged to implement the lifestyle

changes. This group has up to a 25% risk of developing true diabetes within 5

years. If their A1c continues to worsen despite lifestyle intervention, initiation of

metformin prior to actual diagnosis of diabetes can be considered.

The purpose of diabetes treatment is to prevent renal, cardiac, and neurologic

comorbidities, among others. The purpose of prediabetes treatment is to prevent

or at least delay the development of true diabetes. The sooner and more effective

the intervention, the better.

Type 2 diabetes is treated by a combination of lifestyle adjustments and

medications.

Lifestyle

[4] Diet is the most important component of DM management (both overt

diabetes and prediabetics) and usually the hardest way to achieve control. Three

major strategies are used: weight loss, low-fat diet (Ä30% of calories from

fat), and physical exercise. Obese patients should reduce their weight to the ideal

body weight. Metabolic advantages of weight reduction are improved lipid profile

and improved glucose control secondary to increased insulin sensitivity and

decreased insulin resistance. The greater the weight loss, the greater the

improvement in lipid disorders. In the setting of severe obesity (BMI ≥40 or BMI

≥35 with comorbidities), recommendations include consideration of metabolic

surgery (formally called bariatric surgery) (29). [4] Physical exercise promotes

weight loss and improves insulin sensitivity and dyslipidemia in those people who

are in high-risk groups for cardiovascular and microvascular diseases. Treatment

with a statin is recommended in the setting of diabetes to decrease LDL.

Oral Hypoglycemic Agents

Oral hypoglycemic agents are recommended for many type 2 diabetic

patients. The first oral hypoglycemic agents introduced were sulfonylureas (i.e.,

glyburide). The mode of action of sulfonylureas is based on two different

mechanisms: (i) enhanced insulin secretion from the pancreas, and (ii) an

extrapancreatic effect that is poorly understood. Other classes of drugs that have

1180different effects in patients with type 2 diabetes—such as biguanides (metformin),

thiazolidinediones, alpha-glucosidase inhibitors, and insulin secretagogues—were

introduced. Endogenous insulin secretion (as measured by C-peptide) is necessary

for oral hypoglycemic agents to work. If the fasting blood glucose on an adequate

diabetic diet is greater than 250 mg/dL, there is little effect. Frequent evaluation

to monitor control (every 3 to 4 months) is important. If glucose levels cannot be

controlled with oral hypoglycemic agents (i.e., metformin, a biguanide) or other

medicines (i.e., sulfonylureas), insulin therapy should be initiated and referral

should be considered because of the increased rate of complications.

THYROID DISEASES

[5] Thyroid disorders are more common in women and some families,

although the exact rate of inheritance is unknown in geriatric populations,

the incidence may be as high as 5% (31). Thyroid hormones act in target tissues

by binding to nuclear receptors, which induce change in gene expression.

Extrathyroidal conversion of thyroxine (T4) to triiodothyronine (T3) takes place in

the target tissue. T3 binds the nuclear receptor with higher affinity than T4, which

makes T3 more biologically active. Pituitary TSH and hypothalamic thyrotropinreleasing hormone (TRH) regulate hormone production and thyroid growth by

normal feedback physiology. Thyroid-stimulating immunoglobulins (TSI), once

known as a long-acting thyroid stimulator (LATS), bind to the TSH receptor,

which results in the hyperthyroid Graves disease.

More than 99% of circulating T4 and T3 concentrations are bound by

plasma proteins, predominately to thyroxine-binding globulin (TBG), with

the remaining 1% being free. Free levels of thyroid hormones remain constant

despite physiologic or pharmacologic alterations. Regardless of total serum

protein levels, active thyroid hormone levels remain stable. In healthy women,

transitions from puberty to menopause do not alter free thyroid hormone

concentrations. Excess endogenous or exogenous sources of estrogen increase

TBG plasma concentration by decreasing hepatic clearance. Androgens

(especially testosterone) and corticosteroids have the opposite effect by increasing

hepatic TBG clearance.

Thyroid function tests may be misleading in women receiving exogenous

sources of estrogen because of these altered binding characteristics.

Postmenopausal hormonal therapy and pregnancy alter laboratory findings and

complicate interpretation of thyroid function studies. Most laboratories

compensate by reporting a free T4 and T3 level that mathematically corrects for

such physiologic alterations rather than the traditional total T4, and T3 resin

1181uptake (32). Another confounder is that hCG can mimic TSH during the first

trimester of a pregnancy thereby resulting in a falsely low TSH result raising

concerns for hyperthyroidism. If questions arise, a clinical pathologist should be

consulted.

Hypothyroidism

[5] Overt hypothyroidism occurs in 2% of women, and at least an additional

5% develop a laboratory diagnosis of subclinical hypothyroidism.

Hypothyroidism is another disease that disproportionally impacts women five- to

eightfold more commonly than men. The principal cause of hypothyroidism in

countries without iodine deficiencies is autoimmune thyroiditis (Hashimoto

thyroiditis). A familial predisposition is observed in many cases, but the specific

genetic or environmental trigger is unknown. The incidence of autoimmune

thyroiditis increases with age, affecting up to 15% of women older than 65 years

who commonly have only subtle signs or symptoms. [5] Many have “subclinical

hypothyroidism,” which is defined as an elevated serum TSH concentration

with a normal serum free T4 level. It is uncertain whether treatment will

improve the quality of life in otherwise healthy patients who have subclinical

hypothyroidism (31,33). In a setting of autoimmune thyroiditis, one has both

cellular and antibody-mediated destruction of the thyroid, which can result in

either a goiter or atrophic thyroid. Autoimmune thyroiditis may be associated

with other endocrine (e.g., type 1 diabetes, primary ovarian failure, adrenal

insufficiency, and hypoparathyroidism) and nonendocrine (e.g., vitiligo and

pernicious anemia) disorders (33). When any autoimmune disease is diagnosed,

there should be a high degree of suspicion for concurrent thyroid disorders. With

postpartum thyroiditis, there will be a hyperthyroid phase followed by a

hypothyroid phase that can last for months. Iatrogenic causes of hypothyroidism

occur after surgical removal or radioactive iodine therapy for hyperthyroidism

(Graves) or thyroid cancer. Radiation was used to treat acne and other

dermatologic disorders 45 years ago. These patients, now in their 60s or older,

have an increased risk of thyroid cancer and require close monitoring. Although

worldwide iodine deficiency goiter is the most common form of hypothyroidism,

this is uncommon in North America, given the iodine supplementation in salt and

other dietary sources. Hypothyroidism rarely occurs secondary to pituitary or

hypothalamic diseases from TSH or TRH deficiency, but this must be considered

if symptoms occur after neurosurgical procedures.

Clinical Features

Manifestations of hypothyroidism include a broad range of signs and

1182symptoms: fatigue, lethargy, cold intolerance, nightmares, dry skin, hair loss,

constipation, periorbital carotene deposition (causing a yellow discoloration),

carpal tunnel syndrome, weight gain (usually less than 5 to 10 kg),

depression, irritability, hyperlipidemia, and impaired memory. Menstrual

dysfunction is common, either as menorrhagia or amenorrhea. The finding of

hyperlipidemia may be the first indication of hypothyroidism, especially the

presence of high triglycerides. Hypothyroidism may cause precocious or delayed

puberty. Hyperprolactinemia and galactorrhea are unusual manifestations of

hypothyroidism; however, assessment of thyroid function should be considered.

To distinguish primary hypothyroidism from a prolactin-secreting pituitary

adenoma, TSH levels should be assessed in women who have amenorrhea,

galactorrhea, and hyperprolactinemia.

Diagnosis

Recommendations for screening asymptomatic women for thyroid disorders in

women range from every 5 years starting at age 35 in women (American Thyroid

Association), to age 50 (American College of Physicians). Other groups have

recommended periodic screening in older women (American Academy of Family

Physicians and American Association of Clinical Endocrinologists). The USPSTF

stated in their recommendation in 2004 that the evidence is insufficient to

recommend for or against screening (31). In 2014, the USPSTF reviewed the data

regarding routine screening for asymptomatic women without risk factors and

reaffirmed that the evidence is insufficient to recommend for or against screening

(34). [5] For this reason, screening should be reserved for patients at risk (prior

history of thyroiditis or other autoimmune diseases or history of treatment for

hyperthyroidism) or women with symptoms or signs that could represent a

thyroid dysfunction. Suspected hypothyroidism should [5] always be

confirmed with laboratory studies. Primary hypothyroidism is characterized

by the combination of an elevated serum TSH with a low serum free T4 level.

Autoimmune thyroiditis can be confirmed by the presence of serum antithyroid

peroxidase (formerly referred to as antimicrosomal) antibodies. An elevated TSH

with a normal free T4 level implies subclinical hypothyroidism. Central

hypothyroidism, although rare, is distinguished by a low or low-normal serum

free T4 level with either a low or inappropriate normal serum TSH concentration.

Therapy

Synthetic L-thyroxine (T4) is the treatment of choice for hypothyroidism and

is available as generic levothyroxine (35). There is debate about the value of

replacing thyroxine in the subclinical hypothyroidism patient. Such replacement

1183did not result in improved survival, decreased cardiovascular morbidity, or

improve the quality of life (36). The mode of action is by conversion of T4 to T3

in peripheral tissues. Levothyroxine should be taken on an empty stomach.

Absorption may be poor when taken in combination with aluminum hydroxide

(common in antacids), cholestyramine, ferrous sulfate, or fatty meals. The usual

T4 requirement is weight related (approximately 1.6 μg/kg) but decreases for the

elderly. Normal daily dosage is 0.1 to 0.15 mg but should be adjusted to maintain

TSH levels within the normal range. TSH levels should initially be checked in 6

weeks and whenever dosages or brands are changed. When the dose is stabilized,

TSH check once every year or two is adequate unless there is a change in the

patient’s status (i.e., pregnancy).

A low initial T4 dose (0.025 mg per day) should be initiated in the elderly or

patients with known or suspected coronary artery disease. Rapid replacement may

worsen angina and in some cases, induce myocardial infarction.

The use of combined T3 and T4 therapy (desiccated thyroid extracts) is not

recommended for a number of reasons. The conversion of T4 to T3 allows the

normal hormonal regulation to control T3 levels. The use of a combined therapy

overrides that and can result in excessive and nonphysiologic levels of T3

resulting in mild hyperthyroidism. During pregnancy, fetal neurogenesis is

dependent on maternal T4 levels until the estimated gestational age of 16 to 18

weeks (37).

Hyperthyroidism

Hyperthyroidism affects 2% of women during their lifetime, most often

during their childbearing years and impacts women fivefold more commonly

than men. The Graves disease represents the most common disorder; it is

associated with orbital inflammation, causing the classic exophthalmos associated

with the disease and a characteristic dermopathy, pretibial myxedema. It is an

autoimmune disorder caused by TSH reception antibodies that stimulate gland

growth and hormone synthesis. The etiology of the Graves disease in genetically

susceptible women is unknown. Autonomously functioning benign thyroid

neoplasias are less common causes of hyperthyroidism and are associated with

toxic adenomas and toxic multinodular goiter. Transient thyrotoxicosis may be

the result of unregulated glandular release of thyroid hormone in postpartum

(painless, silent, or lymphocytic) thyroiditis and subacute (painful) thyroiditis.

Other rare causes of thyroid overactivity include human chorionic gonadotropin–

secreting choriocarcinoma, TSH-secreting pituitary adenoma, and struma ovarii.

Factitious ingestion or iatrogenic overprescribing should be considered in patients

1184with eating disorders as they use this as a weight control strategy.

Clinical Features

Symptoms of thyrotoxicosis include fatigue, diarrhea, heat intolerance,

palpitations, dyspnea, nervousness, and weight loss. In young patients, there

may be paradoxical weight gain from an increased appetite. Thyrotoxicosis

may cause vomiting in pregnant women, which may be confused with

hyperemesis gravidarum. Tachycardia, lid lag, tremor, proximal muscle

weakness, and warm moist skin are classic physical findings. The most dramatic

physical changes are ophthalmologic and include lid retraction, periorbital edema,

and proptosis. These eye findings occur in less than one-third of women. In

elderly adults, symptoms are often more subtle, with presentations of unexplained

weight loss, atrial fibrillation, or new onset angina pectoris. Menstrual

abnormalities span from regular menses to light flow to anovulatory menses and

associated infertility. Goiter is common in younger women with the Graves

disease, but may be absent in older women. Toxic nodular goiter is associated

with nonhomogeneous glandular enlargement, whereas in subacute thyroiditis the

gland is tender, hard, and enlarged.

Diagnosis

All patients with symptoms of hyperthyroidism should have a complete history

and examination done with focus on the thyroid (nodule, tenderness, or goiter),

cardiac (hypertension tachycardia), pulmonary (tachypnea), neurologic

(peripheral weakness), the eye signs, and presence of peripheral edema or

pretibial myxedema (38).

Most thyrotoxic patients have elevated total and free T4 and T3

concentrations. In thyrotoxicosis, serum TSH concentrations are virtually

undetectable, even with very sensitive assays (sensitivity measured to 0.1 units).

Radioiodine uptake scans are useful in the differential diagnosis of established

hyperthyroidism. Scans with homogeneous uptake of radioactive iodine are

suggestive of the Graves disease, whereas heterogeneous tracer uptake is

suggestive of a diagnosis of toxic nodular goiter. Thyroiditis and medicationinduced thyrotoxicosis have diminished glandular radioisotope concentration.

There is only a modest correlation between the severity of symptoms and the level

of thyroid hormones (38).

Therapy

Therapy can be pharmaceutical, thyroid ablation, thyroidectomy, or a

combination of the three depending on many variables that include the patient’s

age, childbearing plans, and response to other therapies (38).

1185Antithyroid medications, either methimazole (10 to 30 mg per day) or

propylthiouracil (PTU; 50 to 300 mg every 6 to 8 hours) are used for initial

therapy. Both antithyroid drugs block thyroid hormone biosynthesis and may

have additional immunosuppressive effects on the gland. The primary difference

in oral medications is that PTU partially inhibits extrathyroidal T4-to-T3

conversion, whereas methimazole does not. Methimazole has a longer half-life

and permits single daily dosing, which may encourage compliance. Except during

the first trimester of pregnancy when PTU therapy is preferred, methimazole is

the typical first choice in antithyroid medications. Euthyroidism is typically

restored in 3 to 10 weeks, and treatment with oral antithyroid agents is continued

for 6 to 24 months, unless total ablation with radioiodine or surgical resection is

performed. Surgery is less popular because it is invasive and may result in

inadvertent parathyroid removal, which commits the patient to lifelong calcium

therapy.

Beta-adrenergic blocking agents such as propranolol or atenolol are useful

adjunctive therapy for control of sympathomimetic symptoms such as tachycardia

(38). An additional benefit of beta blockers is the blocking of peripheral

conversion of T4 to T3. If a patient is having symptomatic thyrotoxicosis with

heart rate greater than 90 beats per minute or there is a history of pre-existing

cardiovascular disease the patient should be referred to an endocrinologist or even

an emergency room. In rare cases of thyroid storm, PTU, beta blockers,

glucocorticoids, and high-dose iodine preparations (intravenous sodium iodide)

should be administered immediately, and referral to an intensive care unit is

advisable.

The relapse rate with oral antithyroid medications is 50% over a lifetime.

Lifelong follow-up is important when medical therapy is used solely because of

the high relapse rate. Both medications have infrequent (5%) minor side effects,

which include fever, rash, or arthralgias. Major toxicity (e.g., hepatitis, vasculitis,

and agranulocytosis) occurs in less than 1%. PTU appears to be more responsible

for major toxicities than methimazole. Patients on either medication should be

followed with serial complete blood count (CBC) and liver function tests.

However, agranulocytosis cannot be predicted by periodic complete blood counts;

therefore, patients who have a sore throat or fever should stop taking the

medication and call their physician immediately (38).

Therapy with iodine-131 provides a permanent cure of hyperthyroidism in

90% of patients. The principal drawback to radioactive iodine therapy is the high

rate of postablative hypothyroidism, which occurs in at least 50% of patients

immediately after therapy, with additional cases developing at a rate of 2% to 3%

per year. Based on the assumption that hypothyroidism will develop, these

patients should be given lifetime thyroid replacement therapy.

1186Thyroid Nodules and Cancer

[5] Thyroid nodules are common and are more prevalent in adults aged less

than 30 or over 60 years. This is a group that encompasses much of the

population seen by an ob-gyn. For this reason, an understanding of the screening

and diagnosing is important. The vast majority of nodules when discovered by the

patient or the provider, are asymptomatic and benign; however, malignancy (4%

to 6% of all nodules) and hyperthyroidism must be excluded (39). The common

differential includes multinodular goiter, the Hashimoto thyroiditis, colloid/simple

cyst, follicular adenoma, and malignancy. Ultrasound-guided fine-needle

aspiration (FNA) is recommended in the presence of the following factors: history

of radiation to the head, neck, or upper chest; family history of thyroid cancer;

ultrasound findings suggestive of malignancy; or a nodule larger than 1.5 cm in

diameter (40).

Thyroid function tests should be performed before FNA and, if results are

abnormal, the underlying disease should be treated. A markedly suppressed

TSH level implies the nodule is hyperfunctioning and unlikely to be malignant.

Because most nodules are “cold” on scanning (especially if TSH is normal), it is

more cost effective to proceed with ultrasound rather than radioactive scanning.

An ultrasound can determine additional nodules, size of nodule(s), characteristics

of the nodules (solid/cystic), thyroid size, and presence of enlarged lymph nodes.

Thyroid ultrasound findings of solid hypoechoic nodule or features of

microcalcifications, irregular margins, rim calcifications, or evidence of extension

into the surrounding tissue, raise concerns for malignancy. These should be

sampled by FNA irrespective of other findings. The presence of

lymphadenopathy should prompt FNA sampling.

Needle biopsy provides a diagnosis in 95% of cases; in the 5% of patients in

whom the diagnosis cannot be established, excisional biopsy is necessary. Only

20% of excisional biopsies of an “indeterminate aspiration” are found to be

malignant (40). Lesions that are confirmed malignant on biopsy should be treated

with extirpative surgery, and benign nodules should be palpated every 6 to 12

months for growth but surgical intervention is not indicated. Thyroxine

suppressive therapy for benign nodules is not recommended (41).

Papillary thyroid carcinoma is the most common malignancy, found in

75% of thyroid cancers. The majority of cancers are found incidentally during

routine examinations. Risk factors include a history of radiation exposure during

childhood and family history. Signs include rapid growth of neck mass, new onset

hoarseness, or vocal cord paralysis. In the setting of rapid growth, fixed nodule,

new onset hoarseness, or the presence of lymphadenopathy, it is important to be

sure an FNA is done. Thyroidectomy is the primary treatment with radioactive

iodine and TSH suppression with thyroxine. Patients younger than 50 years of age

1187with a primary tumor of less than 4 cm at presentation, even with associated

cervical lymph node metastasis, are usually cured. In the elderly, anaplastic

tumors have a poor prognosis and progress rapidly despite therapy.

Follicular thyroid cancer is the second most common thyroid cancer,

comprising up to 10% of cases. These tend to occur in an older population with

peak ages of 40 to 60. It has a threefold greater prevalence in women than men.

This form of cancer tends to have vascular invasion, frequently with distant

metastases. The prognosis tends to be less favorable with this form of cancer than

with papillary cancers, although women do have a better prognosis than men.

IRRITABLE BOWEL SYNDROME

Irritable bowel syndrome (IBS) is a common problem, affecting about 10% to

15% of the population, with women being twice as likely to have the diagnosis

(42). Given that its primary symptom is typically crampy chronic abdominal pain,

IBS is often in the differential diagnosis for patients with chronic pelvic pain.

Stress and certain foods will often trigger the pain, and defecation often will

provide some relief from the pain. Other gastrointestinal symptoms include

diarrhea and constipation, gastroesophageal reflux disease, nausea, bloating, and

flatulence. What makes this a more difficult diagnosis is the spectrum of

additional symptoms, including dysmenorrhea, dyspareunia, fibromyalgia

complaints, urinary symptoms of frequency and urgency, and even sexual

dysfunction.

This spectrum of symptoms renders diagnosis difficult and led to a consensus

group that created the Rome criteria in 1992, revised in 2005 (43). The resulting

Rome III criteria are: recurrent abdominal pain or discomfort for at least 3 days

per month for 3 months associated with two or more of the following:

Improvement with defecation

Onset associated with a change in the frequency of the stool

Onset associated with a change in the appearance of the stool—

constipation (IBS-C) or diarrhea (IBS-D)

IBS should be a diagnosis of exclusion with consideration initially given to

other causes for the dominant symptom. If that is diarrhea, considerations of

lactose intolerance, infectious etiology, malabsorption, or celiac disease

should be entertained. Symptoms that result in weight loss, rectal bleeding,

anemia, or that are noctural or progressive suggests something other than

IBS unless proven otherwise.

A basic workup might include complete blood count and chemistries.

1188Evaluation of diarrhea, if that is the dominant symptom, should potentially

include stool cultures if infectious etiology is suspected or 24-hour stool

collection (if osmotic) if secretory diarrhea is suspected. Initiate dietary reviews

for lactose intolerance or gluten sensitivity. Flexible sigmoidoscopy/ colonoscopy

is not done routinely unless needed to rule out inflammatory conditions or

malignancy in families with Lynch syndrome or the patient is 50 or older with

sudden onset of symptoms.

Management

General management of IBS can be extremely difficult. Often, the first step is

to reassure the patient that this is a functional disease and is not related to

cancer or malignancy, assuming those were eliminated by history and

examination (44). Many individuals have some underlying concerns that

diagnostic testing needs to be performed or that something is being missed.

Constant reassurance is an important aspect of management. The patient needs to

be an active participant in her care and understand the chronic nature of the

disease. A symptom diary for several weeks may show a link between various

foods and stressors that may be modifiable. Some individuals are able to link

various stressors in their lives to symptoms while others will not have identifiable

causes. Common triggers include stress, anxiety, medication (antibiotics,

antacids), menstrual cycles, abusive relationships, certain foods (lactose,

sorbitol), and travel. Patients should be counseled about dietary

interventions, including increasing dietary fiber, decreasing total fat intake,

and avoiding foods that trigger symptoms. Stool softeners are recommended

for individuals with (IBS-C) hard stools, and bulk aiding agents may be helpful

for those individuals with constipation. The overuse of laxatives is to be

discouraged. Good bowel habits should be discussed. Patients with poor habits

should set aside a quiet time every day to attempt defecation. Many individuals

get into a habit of ignoring stooling symptoms, leading to further problems with

lower gastrointestinal disease.

Antidiarrheal agents, specifically loperamide or diphenoxylate, are often useful

in patients with mild disease with diarrhea as a component (IBS-D). The goal is to

reduce the number of bowel movements and help to relieve rectal urgency.

Anticholinergics including hyoscyamine and dicyclomine hydrochloride often are

helpful. Antispasmodic agents have anticholinergic agents as the primary

ingredient, and compliance may be a problem because side effects include dry

mouth, visual disturbances, and constipation. These agents can precipitate toxic

megacolon, which may result in severe colitis. Toxic megacolon is a medical and

potential surgical emergency, in some cases requiring colectomy. Even though

these patients may be extremely difficult to treat, judicious use of symptom-

1189based pharmacologic approaches (because none have clear benefit),

reassurance, and patient insight may be helpful. The quality of life for some

individuals with IBS is extremely compromised, requiring intense counseling.

It may be difficult to treat them in a busy primary care practice. Those with a

concurrent psychiatric disease, such as depression, will often benefit from

psychiatric consultation and pharmacologic treatment of the underlying disease in

the overall management (45).

Individuals with chronic, debilitating IBS should be referred to a

gastroenterologist. Any suspicion of organic disease with systemic changes,

including weight loss and bloody diarrhea, should be considered for referral.

GASTROESOPHAGEAL REFLUX DISEASE

The term GERD is a commonly used label for many forms of indigestion and

heartburn. The American College of Gastroenterology defines it as

symptoms or mucosal damage produced by the abnormal reflux of gastric

contents into the esophagus (46). The term “abnormal” is key because some

reflux is physiologic, usually occurring postprandial and typically being

asymptomatic. Given the variation in definition, its prevalence is hard to

determine, but it is clear that GERD is more common in the Western world.

Symptoms of GERD include heartburn (burning sensation in the retrosternal

area) commonly postprandial, regurgitation gastric contents into mouth,

dysphagia from esophageal inflammation, and chest pain that can be confused as

angina. The definitive diagnosis of GERD is difficult, so empiric treatment with

acid suppression is reasonable. Dysphagia that is progressive is concerning for

Barrett metaplasia or adenocarcinoma and merits an endoscopic evaluation

(47). Endoscopy should not be used as the first test to diagnose GERD (48).

Treatment of GERD is multifaceted with lifestyle modification and use of

antacids and over-the-counter H2 receptor antagonists or proton pump

inhibitors (PPI) (49). Lifestyle modifications include smoking cessation,

avoidance of eating late in the evening, avoidance of being supine after

eating, weight loss, avoidance of tight clothing, and restriction of alcohol use.

Dietary modifications are helpful but should not be draconian, which will ensure

noncompliance. Key foods to try to minimize are fatty foods, chocolate,

peppermint, and excessive alcohol. The patient can monitor her own symptoms

for the foods that are most problematic for her.

Medications that reduce acid secretions are best and include H2 blockers

or PPIs. They do not prevent the reflux but decrease the damage done by the acid

when refluxed. Medication needs to be titrated to the severity of the symptoms.

H2 blockers commonly work well for acute pain but in placebo-controlled studies

1190in chronic cases without resolution of heartburn after the common 6-week course,

it was found that patients on PPI do better. Maintenance therapy is recommended

for patients who have rapid recurrence of symptoms (in less than 2 to 3 months)

after they stop their medication. Otherwise patients can be managed with episodic

treatments. The linkage of Helicobacter pylori infections and GERD is poorly

understood but seems to be mediated through increased gastric acid

secretion. Treatment can initially worsen GERD and may not improve it (50).

Benefits and risks should be discussed with the patient prior to testing and

treating for H. pylori. The management of GERD during pregnancy is similar to

the treatment in the nonpregnant patient.

CARPAL TUNNEL SYNDROME

Carpal tunnel syndrome (CTS) is the cluster of symptoms brought on by

compression in the carpal tunnel of the median nerve. These are paresthesia,

pain, and weakness. The symptoms are commonly worse at night and may wake

the patient from sleep. It is thought women may be more likely to present with

complaints of CTS because of their small wrists, repetitive motion injury at work

(typing, holding telephone, and reading), and pregnancy with increased edema.

The pain and paresthesia can be located in the wrist or hand or can be in the

forearm. The weakness may cause a patient to have difficulty opening jars, lifting

a plate, turning a doorknob, or holding a glass.

A detailed history is very diagnostic but the use of a couple of simple tests can

help to confirm it (51). The most common one is the Phalen maneuver, in which

the patient flexes her palms at the wrist as close to 90 degrees as possible. Then

with the dorsal portion of the hands touching and the arms parallel to the floor,

the patient presses the flexed hands against each other for approximately 1

minute. This should reproduce her symptoms along the median nerve. The Tinel

test involves percussion over the top of the carpal tunnel where the median nerve

travels. A positive test is when the percussion reproduces the pain and

paresthesia. Additional testing such as nerve conduction studies should be

reserved for patients who do not respond to conservative management or have

significant muscle weakness.

Treatment involves lifestyle modification to decrease repetitive motion

injuries or prolonged marked flexion at the wrist. A carpal tunnel brace can

be very helpful in maintaining adequate extension at the wrist, thereby

“opening” the tunnel and reducing compression on the medial nerve. Only if

these strategies do not work is a surgical intervention indicated.

MITRAL VALVE PROLAPSE SYNDROME, DYSAUTONOMIA,

1191AND POSTURAL ORTHOSTATIC TACHYCARDIA SYNDROME

The terms mitral valve prolapse syndrome (MVPS), dysautonomia, and

postural orthostatic tachycardia syndrome (POTS) all refer to a syndrome in

which the patient has problems with palpitations, hypotension, syncope,

dyspnea, panic/anxiety disorder, numbness, hyperflexible joints, pectus

excavatum, and gastric emptying disorders. Initially patients (typically fivefold

times more likely to be women) who presented with these symptoms were

thought to be somatizing their anxiety disorder. It is now accepted that it is a

syndrome that appears to involve the autonomic nervous system (52). This often

will present first in early adolescence with gradual worsening of the symptoms.

The patients are very slender in build and lose weight to a low body mass index

over a number of months as the syndrome evolves. This weight loss is the

probable cause of the secondary amenorrhea that prompts these women to seek

gynecologic care. The symptoms are not clearly explained by the degree of mitral

valve prolapse, so many feel MVPS is a marker for individuals at risk for this

complex of symptoms. Studies have shown that dysautonomia is an extraarticular

manifestation in the joint hypermobility syndrome (53). Increased sympathetic

activity is the common pathway for most of the proposed mechanisms for POTS

or MVPS. There appears to be a genetic component, with over 10% of patients

reporting the diagnosis in family members with orthostatic intolerance (54). It

needs to be stressed to the patient that the heart is structurally normal.

A tilt table test is often key to the diagnosis. Treatment focuses on the

symptoms and maintaining intravascular volume by encouraging oral intake of

water and salts (55). Physical fitness with aerobic exercises to increase muscle

mass and reduce dependent pooling of blood; avoidance of smoking, caffeine, and

alcohol; and limiting simple carbohydrates will minimize symptoms over time.

Additional medications, including adrenoreceptor agonists, acetylcholinesterase

inhibitor, mineralocorticoid agonist, beta blockers, and selective serotonin

reuptake inhibitors, may be necessary to deal with incompassating symptoms

during the acute phase. Because this is a multifaceted disease, it may be best to

refer the patient during the acute phase to a physician who is experienced with

this syndrome

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